Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1452 |
Axitinib
AG-013736,阿昔替尼,阿西替尼 |
VEGFR; PDGFR; c-Kit | Angiogenesis; Tyrosine Kinase/Adaptors |
Axitinib (AG-013736) 是一种多靶点酪氨酸激酶抑制剂,能够抑制 VEGFR1 (IC50:4 nM),VEGFR2 (IC50:20 nM),VEGFR3 (IC50:0.4 nM),PDGFRβ (IC50:2 nM)。 | |||
T21129 |
Axitinib sulfoxide
Axitinib metabolite M12,PF-03482595,AG-028458 |
||
Axitinib sulfoxide is a major metabolite of Axitinib, which is a VEGFR tyrosine kinase inhibitor and may be useful in cancer therapy. |