Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2753 |
Avasimibe
PD-148515,阿伐麦布,CI-1011 |
P450; Acyltransferase | Metabolism |
Avasimibe (PD-148515) 是一种口服有效的酰基辅酶 A: 胆固醇酰基转移酶 (ACAT) 抑制剂,对 ACAT1和 ACAT2的 IC50分别为 24 和 9.2 µM。Avasimibe 在前列腺癌中有研究的价值。 | |||
T70300 |
Avasimibe sodium
|
||
Avasimibe sodium is an acyl coenzyme A: cholesterol acyltransferase (ACAT) inhibitor. | |||
T70299 | PF-05214030 | ||
PF-05214030 is a novel potent TRPV4 antagonist (hTRPV4 IC50 4nM; rTRPV4 IC50 27nM). |