Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1223 |
Apamin
Apamine |
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Apamin (Apamine) is an 18 amino acid peptide neurotoxin found in apitoxin (bee venom), is known as a specifically selective blocker of Ca2+-activated K+ (SK) channels and exhibits anti-inflammatory and anti-fibrotic activity. Apamin is a bee venom compone | |||
TP1223L |
Apamin acetate
Apamine acetate,Apamin acetate(24345-16-2 Free base) |
Potassium Channel | Membrane transporter/Ion channel |
Apamin acetate (Apamine acetate) 是一种具有选择性的 Ca2+ 激活的 K+ (SK) 通道的阻断剂,是在蜂毒素中发现的一种 18 个氨基酸的肽类神经毒素。Apamin acetate 可增强皮质神经元撕裂损伤后的神经突生长和再生。Apamin acetate 具有抗炎和抗纤维化的作用。 | |||
TP1222 |
Apamin TFA (24345-16-2 free base)
Apamin TFA,Apamine TFA |
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Apamin TFA (Apamine TFA) is a toxin found in bee venom. It is a potent blocker of small conductance Ca2+-activated K+ (SK, KCa2) channels that is more effective at SK2 than SK1 and SK3. | |||
T75746 |
Apamin TFA
|
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Apamin TFA (Apamine TFA) 是在蜂毒素中发现的一种 18 个氨基酸的肽类神经毒素,是一种 Ca2+激活的 K+(SK) 通道的特异性和选择性的阻断剂,具有抗炎和抗纤维化的作用。 | |||
T20968 |
CyPPA
|
Potassium Channel; Dopamine Receptor | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
CyPPA 是hSK2和hSK3的阳性调节剂,其EC50值分别为 5.6 μM 和14 μM。它对 hSK1 和 hIK 通道无活性。 | |||
T0979 |
Dequalinium chloride
Dequafungan,地喹氯铵,Danical,Decabis |
Potassium Channel; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel |
Dequalinium chloride (Decabis) 是一种apamin 敏感型的钾离子通道选择性阻断剂。 | |||
T23493 |
UCL 1684 dibromide
UCL 1684 |
Others | Others |
apamin-sensitive Ca2+-activated K+ channel (KCa2.1) blocker | |||
TMIH-0183 |
Dequalinium Chloride-d4
|
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Dequalinium Chloride-d4 是 Dequalinium Chloride 的氘代化合物。Dequalinium Chloride 的 CAS 号为 522-51-0。Dequalinium chloride 是一种apamin敏感型的钾离子通道选择性阻断剂。 |