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Cat. No. Product Name Target Signaling Pathways
T7743 ANGIOTENSIN IV TFA(12676-15-2(free base))

RAAS Endocrinology/Hormones
ANGIOTENSIN IV TFA(12676-15-2(free base)) 是一种不太有效的血管紧张素 AT1 受体激动剂。
T5824 Angiotensin II (3-8), human

Angiotensin IV

RAAS Endocrinology/Hormones
Angiotensin II (3-8), human 是活性稍弱的血管紧张素AT1受体激动剂。
T7376 Dihexa

PNB-0408,Hexanoyl-Tyr-Ile-Ahx-NH2,N-hexanoic-Try-Ile-(6)-amino hexanoic amide

c-Met/HGFR Tyrosine Kinase/Adaptors
Dihexa (Hexanoyl-Tyr-Ile-Ahx-NH2) 是肝细胞生长因子/c-Met (HGF/c-Met) 系统的激活剂,它与 HGF (Kd = 65 pM) 结合,是肽血管紧张素 IV 的类似物。
T70932 L6H9

L6H9 is a novel inhibitor of myeloid differentiation factor 2 (MD2), suppressing HG-induced expression of ACE and AT1 receptor and Angiotensin II (AngII) production in renal NRK‐52E cells, resulting in the decrease in fibrosis markers such as TGF-β and collagen IV.
TP1404 Hemorphin-7

Hemorphin-7 binds to the angiotensin IV receptor, triggering multiple effects including cellular proliferation and memory enhancement. Hemorphins are endogenous peptides belonging to the family of atypical opioid peptides released from hydrolyzed hemoglob
TP1990 Norleual

Angiotensin IV analog. Highly potent HGF/c-MET inhibitor (IC50 = 3 pM). Inhibits HGF-induced MDCK cell proliferation and invasion in vitro. Also AT4 receptor antagonist; disrupts LTP stabilization. Antiangiogenic.
T75940 Norleual TFA

Norleual TFA 是一种血管紧张素 (Ang) IV 类似物,是一种肝细胞生长因子(HGF)/c-Met 抑制剂,IC50为 3 pM。Norleual TFA 还是一种AT4拮抗剂,具有强大的抗血管生成活性。

化合物

ANGIOTENSIN IV TFA(12676-15-2(free base))
Cat.No: T7743
Synonym:
Target: RAAS
Angiotensin II (3-8), human
Cat.No: T5824
Synonym: Angiotensin IV
Target: RAAS
Dihexa
Cat.No: T7376
Synonym: PNB-0408,Hexanoyl-Tyr-Ile-Ahx-NH2,N-hexanoic-Try-Ile-(6)-amino hexanoic amide
Target: c-Met/HGFR
L6H9
Cat.No: T70932
Synonym:
Target:
Hemorphin-7
Cat.No: TP1404
Synonym:
Target:
Norleual
Cat.No: TP1990
Synonym:
Target:
Norleual TFA
Cat.No: T75940
Synonym:
Target:
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