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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T1454 Acyclovir

Aciclovir,Acycloguanosine,阿昔洛韦

Apoptosis; DNA/RNA Synthesis; Antibacterial; Antibiotic; HSV Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Acyclovir (Aciclovir) 是鸟嘌呤类似物和具有口服活性的抗病毒剂。它对HSV-1(IC50为 0.85 μM),HSV-2(IC50为 0.86 μM) 和水痘带状疱疹病毒有活性。
T20406 Acyclovir L-isoleucinate

Acyclovir isoleucinate

Acyclovir L-isoleucinate is an acyclovir impurity. It also is an Acyclovir amino acid ester prodrug.
T23626 Acyclovir alaninate

Acyclovir alanine is a pro-drug of Acyclovir. Acyclovir works by decreasing the production of DNA of the virus and it shows very low cytotoxicity.
T1454L Acyclovir sodium

Aciclovir sodium

Acyclovir sodium is an antimetabolite. Acyclovir sodium inhibits HSV-specified DNA polymerases and prevents further viral DNA synthesis.
T29628 Acyclovir mixture with hydrocortisone

Xerese,ME 609,ME609,ME-609,Lipsovir

Acyclovir mixture with hydrocortisone is used for Herpes simplex labialis.
T60709 Acyclovir monophosphate

Acyclovir monophosphate 是抗单纯疱疹病毒 (HSV)剂,并且具有抗肿瘤活性。Acyclovir monophosphate 通过抑制病毒 DNA 聚合酶从而阻断 DNA 合成,同时能终止病毒 DNA 的链延伸。
T22304 Desciclovir

BW A515U,地昔洛韦,6-Deoxyacyclovir,DCV

Antifection Microbiology/Virology
Desciclovir (DCV) 是抗疱疹药物阿昔洛韦的前药,口服有活性,在体内被黄嘌呤氧化酶转化成为阿昔洛韦。
T1087 Valacyclovir hydrochloride

Valaciclovir hydrochloride,盐酸伐昔洛韦,盐酸万乃洛韦,Valaciclovir HCl

DNA/RNA Synthesis; Antibiotic; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Valacyclovir hydrochloride (Valaciclovir hydrochloride) 是一种口服有效的抗病毒药物,能抑制疱疹 B,单纯疱疹和带状疱疹。它抑制 HSV-1W,IC50为2.9 μg/ml。它是 Aciclovir 的前药。
T64299 Valacyclovir hydrochloride hydrate

Valacyclovir hydrochloride hydrate 是一种有效的抗病毒剂,是一种前药,在体内可快速转化为阿昔洛韦。Valacyclovir hydrochloride hydrate 能够用于配制治疗眼部疱疹的眼部插入物。Valacyclovir hydrochloride hydrate 能够用于单纯疱疹、带状疱疹和乙型疱疹的治疗。
T20927 Benzyloxycarbonyl valacyclovir

Benzyloxycarbonyl valacyclovir is a biochemical.
T35010 Valacyclovir Related Compound D

N-Ethyl valacyclovir

Valacyclovir Related Compound D is a bioactive chemical.
T65324 Diacetylacyclovir

Diacetylacyclovir 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65324,CAS号为 75128-73-3。
T0688 Ganciclovir

BW 759,更昔洛韦,RS-21592,2'-Nor-2'-deoxyguanosine

Nucleoside Antimetabolite/Analog; Others; Antibiotic; Antifection; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Ganciclovir (2'-Nor-2'-deoxyguanosine) 是核苷类似物和口服抗病毒药物,对CMV 具有抗病毒活性。它用于治疗与艾滋病相关的巨细胞病毒感染的并发症。
T31659 Eprociclovir

AV10,AV-10,A-5021,A 5021,A5021,AV 10

Antifection Microbiology/Virology
Eprociclovir (A-5021) 是一种新型阿昔洛韦类似物,是 EHV1 复制的强效抑制剂,可能用于治疗和/或预防该病毒感染。Eprociclovir 对大多数人类疱疹病毒都有很强的抗疱疹活性。
T70027 Eprociclovir potassium

Eprociclovir potassium is a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applied onto the affected cornea, ameliorated clinica...
T69817 Eprociclovir Na

Eprociclovir Na is the salt form of Eprociclovir, also known as A-5021, a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applie...
T40911 9-Carboxymethoxymethylguanine

9-Carboxymethoxymethylguanine is the primary metabolite derived from Aciclovir, a guanosine analogue with potent antiviral properties. Aciclovir, also known as Acyclovir, acts as an orally active antiviral agent.
T68957 Eprociclovir dihydrate

Eprociclovir dihydrate is a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applied onto the affected cornea, ameliorated clinica...
T36490 AZT triphosphate TEA

AZT triphosphate TFA (3'-Azido-3'-deoxythymidine-5'-triphosphate TFA) is a active triphosphate metabolite of Zidovudine (AZT). AZT triphosphate TFA exhibits antiretroviral activity and inhibits replication of HIV. AZT triphosphate TFA also inhibits the DNA polymerase of HBV. AZT triphosphate TFA activates the mitochondria-mediated apoptosis pathway[1][2][3]. Treatment with 100 μM Zidovudine (AZT) for 48h disrupts the mitochondrial tubular network via accumulation of AZT triphosphate (AZT-TP) in ...

化合物

Acyclovir
Cat.No: T1454
Synonym: Aciclovir,Acycloguanosine,阿昔洛韦
Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic, HSV
Acyclovir L-isoleucinate
Cat.No: T20406
Synonym: Acyclovir isoleucinate
Target:
Acyclovir alaninate
Cat.No: T23626
Synonym:
Target:
Acyclovir sodium
Cat.No: T1454L
Synonym: Aciclovir sodium
Target:
Acyclovir mixture with hydrocortisone
Cat.No: T29628
Synonym: Xerese,ME 609,ME609,ME-609,Lipsovir
Target:
Acyclovir monophosphate
Cat.No: T60709
Synonym:
Target:
Desciclovir
Cat.No: T22304
Synonym: BW A515U,地昔洛韦,6-Deoxyacyclovir,DCV
Target: Antifection
Valacyclovir hydrochloride
Cat.No: T1087
Synonym: Valaciclovir hydrochloride,盐酸伐昔洛韦,盐酸万乃洛韦,Valaciclovir HCl
Target: DNA/RNA Synthesis, Antibiotic, HSV
Valacyclovir hydrochloride hydrate
Cat.No: T64299
Synonym:
Target:
Benzyloxycarbonyl valacyclovir
Cat.No: T20927
Synonym:
Target:
Valacyclovir Related Compound D
Cat.No: T35010
Synonym: N-Ethyl valacyclovir
Target:
Diacetylacyclovir
Cat.No: T65324
Synonym:
Target:
Ganciclovir
Cat.No: T0688
Synonym: BW 759,更昔洛韦,RS-21592,2'-Nor-2'-deoxyguanosine
Target: Nucleoside Antimetabolite/Analog, Others, Antibiotic, Antifection, HSV
Eprociclovir
Cat.No: T31659
Synonym: AV10,AV-10,A-5021,A 5021,A5021,AV 10
Target: Antifection
Eprociclovir potassium
Cat.No: T70027
Synonym:
Target:
Eprociclovir Na
Cat.No: T69817
Synonym:
Target:
9-Carboxymethoxymethylguanine
Cat.No: T40911
Synonym:
Target:
Eprociclovir dihydrate
Cat.No: T68957
Synonym:
Target:
AZT triphosphate TEA
Cat.No: T36490
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN3559 Cabraleahydroxylactone

HSV Microbiology/Virology
Cabraleahydroxylactone displays antimycobacterial activity against Mycobacterium tuberculosis, it is weakly cytotoxic to a breast cancer (BC) cell line.It shows antiviral activity against herpes simplex virus type-1 with an IC50 value of 3.20 ug/mL, in comparison with the standard acyclovir (IC50=1.90ug/mL).

天然产物

Cabraleahydroxylactone
Cat.No: TN3559
Synonym:
Target: HSV
TargetMol Loading
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