Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6078 |
Saracatinib
AZD0530,塞卡替尼 |
EGFR; Src; BTK; Autophagy | Angiogenesis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Saracatinib (AZD0530) 是一种有效的 Src 抑制剂,抑制 c-Src、Lck、c-YES、Lyn、Fyn、Fgr 和 Blk 的 IC50值在 2.7 到 11 nM 之间,对其他酪氨酸激酶具有选择性。 | |||
T68425 |
Saracatinib difumarate
|
||
Saracatinib difumarate is an orally available dual-specific inhibitor of Src and Abl with anti-invasive and anti-tumor activities. |