Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T41190 |
AY 77
Unk-Cha-Chg-NH2 |
ERK; Calcium Channel; Protease-activated Receptor | GPCR/G Protein; MAPK; Membrane transporter/Ion channel; Metabolism |
AY 77 (Unk-Cha-Chg-NH2)是一种有效的、具有选择性的 PAR2激动剂。AY 77对 Ca2+和 ERK1/2信号显示出选择性(Ca2+释放的ec50值为40 nM, ERK1/2磷酸化的ec50值为2 μM)。AY 77能够促进人乳腺癌细胞的体外迁移。 |