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Cat. No. Product Name Target Signaling Pathways
T23653 Afegostat HCl

Afegostat,AT-2101,Afegostat hydrochloride,AT2101

Afegostat is an acid β-glucosidase (GCase) active site inhibitor that acts as a pharmacological chaperone. Afegostat inhibits GCase with K(i) ~30 nM for wild-type and mutant enzymes. Afegostat was an experimental drug for the treatment of certain forms of
T71474 H-201-70

H-201-70 is a partial beta1 agonist with adrenoreceptor stimulatory effects.
T28424 PKUMDL-WQ-2101

Dehydrogenase Metabolism
PKUMDL-WQ-2101 是磷酸甘油酸脱氢酶的选择性变构抑制剂,具有抗肿瘤活性。
TP2101 Z-VRPR-FMK trifluoroacetate salt

Irreversible MALT1 inhibitor. Suppresses T cell activation-induced cleavage of Bcl-10 in a dose-dependent manor. Reduces Jurkat cell adhesion to fibronectin. Cell permeable.

化合物

Afegostat HCl
Cat.No: T23653
Synonym: Afegostat,AT-2101,Afegostat hydrochloride,AT2101
Target:
H-201-70
Cat.No: T71474
Synonym:
Target:
PKUMDL-WQ-2101
Cat.No: T28424
Synonym:
Target: Dehydrogenase
Z-VRPR-FMK trifluoroacetate salt
Cat.No: TP2101
Synonym:
Target:
TargetMol Loading
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