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Targets Recommended: PARP

4

抑制剂 & 化合物

2

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T72553 ARTD10/PARP10-IN-1

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
ARTD10/PARP10-IN-1 是一种强效性的 PARP 抑制剂,抑制单 ADP 核糖转移酶 ARTD7/PARP15,ARTD8/PARP14,ARTD10/PARP10 和聚 ADP-核糖聚合酶-1 (ARTD1/PARP1),具有潜在的抗癌抗肿瘤活性,可用于研究前列腺癌和乳腺癌。
T72554 ARTD10/PARP10-IN-2

ARTD10/PARP10-IN-2 是一种强效、非选择性的PARP 抑制剂。ARTD10/PARP10-IN-2 靶向单 ADP 核糖转移酶 (ARTD10/PARP10) 和聚 ADP-核糖聚合酶-1 (ARTD1/PARP1),IC50分别为 2.0 μM,和 9.7 μM。
T3168 MN-64

MN64

Others; PARP; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Others; Stem Cells
MN-64 是一种有效的tankyrase 1抑制剂,对TNKS1、TNKS2、ARTD1ARTD2 的IC50值分别为 6、72、19.1 和 39.4 μM。
T11143 EB-47

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
EB-47 是一种有效的 PARP-1/ARTD-1 选择性抑制剂,IC50 值为 45 nM,对 ARTD5 的IC50 值为 410 nM,表现出温和的药效。EB-47 模拟底物 NAD+,从烟酰胺延伸至腺苷亚区结合。

化合物

ARTD10/PARP10-IN-1
Cat.No: T72553
Synonym:
Target: PARP
ARTD10/PARP10-IN-2
Cat.No: T72554
Synonym:
Target:
MN-64
Cat.No: T3168
Synonym: MN64
Target: Others, PARP, Wnt/beta-catenin
EB-47
Cat.No: T11143
Synonym:
Target: PARP
Cat. No. Product Name Species Expression System
TMPY-01188 PARP Protein, Human, Recombinant (His)

ADPRT1,ADPRT,pADPRT-1,PPOL,ARTD

Human Baculovirus Insect Cells
PARP Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 114.5 kDa and the accession number is A0A024R3T8.
TMPY-02465 PARP Protein, Mouse, Recombinant (His)

AI893648,Adprp,5830444G22Rik,C80510,sPARP-1

Mouse Baculovirus Insect Cells
PARP Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 115 kDa and the accession number is Q921K2.

重组蛋白

PARP Protein, Human, Recombinant (His)
Cat.No: TMPY-01188
Species: Human
Expression System: Baculovirus Insect Cells
PARP Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02465
Species: Mouse
Expression System: Baculovirus Insect Cells
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