Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2466 |
Osu03012
Osu-03012,Osu 03012,AR-12 |
PDK | PI3K/Akt/mTOR signaling |
Osu03012 (AR-12) 是一种口服生物可利用的小分子塞来昔布衍生的磷酸肌醇依赖性激酶 1(PDK1) 抑制剂,具有潜在的抗肿瘤活性。 | |||
T5677 |
SAR125884 hydrochlorid (1116743-46-4(free base))
|
c-Met/HGFR | Tyrosine Kinase/Adaptors |
SAR125884 hydrochlorid (1116743-46-4(free base)) 是一种有效的选择性 MET 激酶抑制剂,具有良好的临床前毒性特征 (IC50=4.2 nM)。 | |||
T5467 |
SAR125844
SAR125884 |
Apoptosis; c-Met/HGFR | Apoptosis; Tyrosine Kinase/Adaptors |
SAR125844 是高度选择性可逆ATP 竞争性的MET 受体酪氨酸激酶抑制剂,其IC50值为4.2 nM。能抑制细胞中MET 的自磷酸化。 | |||
T24758 |
SAR127303
SAR-127303,SAR 127303 |
||
SAR127303 is an effective covalent inhibitor of MAGL. SAR127303 behaves as a selective and competitive inhibitor of mouse and human MAGL. |