Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0811L |
Amisulpride hydrochloride
APD-421,Amisulpride HCl,APD 421,APD421,Sultopride,氨磺必利盐酸盐 |
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Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth. | |||
T7180L |
Sultopride
舒托必利,LIN1418,LIN-1418,Sultopridum,LIN 1418 |
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Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group. | |||
T26375 |
(S)-Amisulpride
Esamisulpride,(S) Amisulpride,SEP-4199,(S)-氨磺必利 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
(S)-Amisulpride ((S) Amisulpride) 是一种有效的多巴胺D2/D3受体拮抗剂,具有抗精神和抗抑郁作用。它是5-HT7受体的拮抗剂,KI 值为 900 nM。 | |||
T0811 |
Amisulpride
DAN 2163,氨磺必利,阿米舒必利 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Amisulpride (DAN 2163) 是多巴胺D2/D3受体拮抗剂,对于人多巴胺D2和D3的Ki 分别为 2.8 和 3.2 nM。 |