Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2641 |
KRCA-0008
KRCA 0008,KRCA0008 |
ACK; ALK | Angiogenesis; Tyrosine Kinase/Adaptors |
KRCA-0008 是高效的、选择性的 ALK/Ack1 抑制剂,对ALK 和Ack1的IC50值分别为12nM 和4nM,显示出非hERG 依赖性药物活性。 | |||
T21361 |
Alclometasone dipropionate
Vaderm,Sch 22219,Aclovate,Delonal |
Others | Others |
Alclometasone dipropionate (Sch 22219) 是一种人工合成的糖皮质激素,属于类固醇化合物,具有抗增生、抗炎、抗过敏、止痒和收缩血管的作用,可用于研究皮肤炎症。 | |||
T29842 |
Alclofenac
W 7320,烯氯苯乙酸,MY 101,BRN 2116510,W-7320,W7320 |
Others | Others |
Alclofenac (W-7320) 对急性期蛋白反应和L-色氨酸与血浆蛋白结合程度有显著影响,可用于慢性风湿病患者的治疗。 | |||
T14154 |
Alclometasone
7a-Chloro-16a-methyl prednisolone |
||
Alclometasone (7a-Chloro-16a-methyl prednisolone), a glucocorticoid, inhibits leukocytes from releasing pro-inflammatory mediators. It is effective in treating corticosteroid-responsive dermatoses such as atopic dermatitis, psoriasis, allergic dermatitis, and eczema [1]. | |||
T35012 | Valclavam | ||
Valclavam is a biochemical. | |||
T25036 | Alclofenac sodium | ||
Alclofenac sodium is an anti-inflammatory utilized in the treatment of rheumatoid arthritis. | |||
T25035 |
Alclofenac lysinate
|
||
Alclofenac is an anti-inflammatory agent used in the treatment of rheumatoid arthritis. It also used as an analgesic and an antipyretic. | |||
T29843 |
Alcloxa
RC-173,RC 173 |
||
Alcloxa is a astrigent. | |||
T2251 |
NVP-TAE 684
TAE684,5-氯-N2-[2-甲氧基-4-[4-(4-甲基-1-哌嗪基)-1-哌啶基]苯基]-N4-[2-[(1-甲基乙基)磺酰基]苯基]-2,4-嘧啶二胺 |
Apoptosis; ALK | Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors |
NVP-TAE 684 (TAE684) 是一种高效特异性 ALK 抑制剂,阻止 ALCL 衍生的 ALK 依赖性细胞株的生长,IC50值为 3 nM。 | |||
T77041 | Iratumumab | ||
Iratumumab (MDX-060),一种人来源IgG1κ型CD30单克隆抗体,能够抑制表达CD30的肿瘤细胞生长。适用于霍奇金淋巴瘤(HL)与间变性大细胞淋巴瘤(ALCL)的研究。 |