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Cat. No. Product Name Target Signaling Pathways
T3467 Miransertib

ARQ-092,AKT inhibitor 2

Akt; Parasite Cytoskeletal Signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling
Miransertib (ARQ-092) 是一种具有口服活性的,选择性和变构性Akt 抑制剂。它有效抑制利什曼原虫,还是 AKT1-E17K 突变蛋白抑制剂,可研究PI3K/AKT 驱动的肿瘤和 Proteus 综合征。
T38846 Vevorisertib trihydrochloride

ARQ 751 trihydrochloride

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Vevorisertib trihydrochloride(ARQ 751 trihydrochloride) 是一种具有选择性和有效性的 pan-AKT 和 AKT1-E17K 突变抑制剂,抑制 AKT1AKT2 和 AKT3 。 Vevorisertib trihydrochloride 可用于研究肝癌和晚期实体瘤。
T22247 Miransertib (ARQ 092) HCl

Miransertib hydrochloride (ARQ-092 hydrochloride) is a powerful, orally bioavailable, selective, and allosteric inhibitor of Akt. It exhibits an inhibitory concentration (IC50) of 2.7 nM, 14 nM, and 8.1 nM against Akt1, Akt2, and Akt3, respectively. In addition to its Akt inhibitory activity, Miransertib hydrochloride also demonstrates significant potency as an inhibitor of the AKT1-E17K mutant protein. This compound shows promise in research related to PI3K/AKT-driven tumors and Proteus syndrom...

化合物

Miransertib
Cat.No: T3467
Synonym: ARQ-092,AKT inhibitor 2
Target: Akt, Parasite
Vevorisertib trihydrochloride
Cat.No: T38846
Synonym: ARQ 751 trihydrochloride
Target: Akt
Miransertib (ARQ 092) HCl
Cat.No: T22247
Synonym:
Target:
TargetMol Loading
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