Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2047 |
AG-1478
AG1478,NSC 693255,Tyrphostin AG-1478 |
EGFR; HCV Protease; Influenza Virus; HER; PDGFR | Angiogenesis; JAK/STAT signaling; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors |
AG-1478 (NSC-693255) 是一种选择性 EGFR 酪氨酸激酶抑制剂,IC50为 3 nM。它对 HCV 和脑心肌炎病毒有抗病毒作用。 | |||
T20199 |
AG-1478 hydrochloride
AG1478 HCl,AG-1478 HCl,Tyrphostin,AG1478 Hydrochloride,AG 1478 HCl |
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AG1478 HCl is an epidermal growth factor receptor protein inhibitor. | |||
T27787L |
L-797,591 hydrochloride
L-797,591 hydrochloride(217480-24-5 Free base) |
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L-797,591 hydrochloride 对生长抑素受体亚型 1 (SSTR1)有活性。L-797,591 hydrochloride 常与 AG1478 联合使用来增强表达 SSTR1的细胞中 p-ERK5的表达。L-797,591 hydrochloride 在共转染的细胞中显著增强了 p38的磷酸化,这一作用在与 AG1478联合处理时被逆转。 |