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7

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T40872 17-AEP-GA

17-AEP-GA is a highly effective HSP90 antagonist compound that exhibits potent inhibition against the proliferation, survival, migration, and invasion of glioblastoma cells. Additionally, it demonstrates ADCs Toxin activity.
T61004 AEP-IN-1

APE-IN-1 可用于阿尔茨海默病的早期诊断和药物研发。APE-IN-1 是一种有效的天冬酰胺内肽酶(APE) 抑制剂,IC50值为 89 nM。
T9713 δ-secretase inhibitor 11

Beta Amyloid; Caspase Apoptosis; Neuroscience; Proteases/Proteasome
δ-secretase inhibitor 11是一种分泌酶抑制剂,可用作 阿尔茨海默病(AD) 治疗转化开发的先导化合物。
T18304 Mal-VC-PAB-ABAEP-Azonafide

Others Others
Mal-VC-PAB-ABAEP-Azonafide, an ADC (antibody-drug conjugate) linker-drug conjugate, demonstrates potent antitumor activity. It incorporates Azonafide, a cytotoxin, connected through the ADC linker Mal-VC-PAB[1].
T33578 Naepaine hydrochloride

Naepaine hydrochloride is a biochemical.
T25847 NAEPA

NAEPA, an LPA mimetic, is a selective agonist of the lysophosphatidic acid-1 (LPA1) receptor.
T38116 Fmoc-Ala-Glu-Asn-Lys-NH2

Fmoc-Ala-Glu-Asn-Lys-NH2

Fmoc-Ala-Glu-Asn-Lys-NH2 is a peptide inhibitor that selectively targets asparagine endopeptidase (AEP) and inhibits the cleavage of amyloid precursor protein (APP). AEP, a pH-controlled cysteine proteinase, plays a crucial role in the proteolytic processing of APP, and its activity is enhanced during the aging process [1].

化合物

17-AEP-GA
Cat.No: T40872
Synonym:
Target:
AEP-IN-1
Cat.No: T61004
Synonym:
Target:
δ-secretase inhibitor 11
Cat.No: T9713
Synonym:
Target: Beta Amyloid, Caspase
Mal-VC-PAB-ABAEP-Azonafide
Cat.No: T18304
Synonym:
Target: Others
Naepaine hydrochloride
Cat.No: T33578
Synonym:
Target:
NAEPA
Cat.No: T25847
Synonym:
Target:
Fmoc-Ala-Glu-Asn-Lys-NH2
Cat.No: T38116
Synonym: Fmoc-Ala-Glu-Asn-Lys-NH2
Target:
Cat. No. Product Name Target Signaling Pathways
T4703 (2-Aminoethyl)phosphonic acid

2-Aminoethylphosphonic acid,2-氨基乙基膦酸,Ciliatine,2-AEP

Others; Endogenous Metabolite Metabolism; Others
(2-Aminoethyl)phosphonic acid (2-Aminoethylphosphonic acid) 主要在尿液中检测到。(2-Aminoethyl)phosphonic acid 参与许多酶促反应,也是其他转化产物的母体化合物,包括但不限于神经酰胺 2-(甲氨基)乙基膦酸酯、N-(2-膦乙基)胆酰胺和 CMP-2-氨基乙基膦酸酯。

天然产物

(2-Aminoethyl)phosphonic acid
Cat.No: T4703
Synonym: 2-Aminoethylphosphonic acid,2-氨基乙基膦酸,Ciliatine,2-AEP
Target: Others, Endogenous Metabolite
TargetMol Loading
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