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Cat. No. Product Name Target Signaling Pathways
T15384 Glesatinib

MGCD265

c-Met/HGFR Tyrosine Kinase/Adaptors
Glesatinib is an orally active and potent dual inhibitor of MET/SMO. Glesatinib is also a tyrosine kinase inhibitor. It antagonizes P-glycoprotein mediated multidrug resistance (MDR) in NSCLC.
T6351 MGCD-265 analog

MGCD-265,Glesatinib

Apoptosis; VEGFR; c-Met/HGFR Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
MGCD-265 analog (Glesatinib) 是一种口服生物可利用的多靶点酪氨酸激酶抑制剂,具有抗肿瘤活性,对 c-Met 和 VEGFR2 的 IC50 分别为 29 nM 和 10 nM。
T15383 Glesatinib hydrochloride

MGCD265 hydrochloride

c-Met/HGFR Tyrosine Kinase/Adaptors
Glesatinib hydrochloride is an orally active and potent dual inhibitor of MET/SMO. Glesatinib hydrochloride is also a tyrosine kinase inhibitor. It antagonizes P-glycoprotein mediated multidrug resistance (MDR) in NSCLC.

化合物

Glesatinib
Cat.No: T15384
Synonym: MGCD265
Target: c-Met/HGFR
MGCD-265 analog
Cat.No: T6351
Synonym: MGCD-265,Glesatinib
Target: Apoptosis, VEGFR, c-Met/HGFR
Glesatinib hydrochloride
Cat.No: T15383
Synonym: MGCD265 hydrochloride
Target: c-Met/HGFR
TargetMol Loading
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