Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6081 |
Milciclib
PHA-848125 |
Trk receptor; CDK; Autophagy | Autophagy; Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors |
Milciclib (PHA-848125) 是一种 ATP 竞争性的 CDK 和原肌球蛋白受体激酶双重抑制剂,作用于 CDK2,IC50 为 45 nM。 | |||
T71121 |
Milciclib maleate
|
||
Milciclib maleate is an inhibitor of cyclin-dependent kinases (CDKs) and thropomyosin receptor kinase A (TRKA). |