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Cat. No. Product Name Target Signaling Pathways
TN2883 3',4'-Dimethoxyflavone

Others; PARP Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
3',4'-Dimethoxyflavone 是类黄酮化合物的参考标准,类黄酮化合物具有多种药用活性。
TN5133 3',5,5',7-Tetrahydroxy-4',6-dimethoxyflavone

HIV Protease; Topoisomerase DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
5,7,3',5'-tetrahydroxy-6,4'-dimethoxyflavone exhibits anti-HIV-1 activity in the anti-syncytium assay using (∆Tat/rev)MC99 virus and 1A2 cell line system, it shows considerably activity against HIV-1 reverse transcriptase. It exhibits cytotoxic activity against P-388 cell lines, it can inhibit DNA topoisomerase IIα activity, which may be responsible for the observed cytotoxicity.

天然产物

3',4'-Dimethoxyflavone
Cat.No: TN2883
Synonym:
Target: Others, PARP
3',5,5',7-Tetrahydroxy-4',6-dimethoxyflavone
Cat.No: TN5133
Synonym:
Target: HIV Protease, Topoisomerase
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