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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T37955 Sphingosine-1-phosphate (d16:1)

Sphingosine-1-phosphate (d16:1)

C16 Sphingosine-1-phosphate (C16 S1P) is a derivative of sphingosine-1-phosphate that binds to S1P1/EDG-1, S1P3/EDG-3, and S1P2/EDG-5 receptors with affinities of 115%, 83%, and 103%, respectively, relative to S1P in CHO cells. C16 S1P was increased in postmortem primary open angle glaucoma trabecular meshwork samples.

化合物

Sphingosine-1-phosphate (d16:1)
Cat.No: T37955
Synonym: Sphingosine-1-phosphate (d16:1)
Target:
Cat. No. Product Name Target Signaling Pathways
T21500 Sphingosine-1-phosphate

S1P

Endogenous Metabolite; S1P Receptor; LPL Receptor GPCR/G Protein; Metabolism
Sphingosine-1-phosphate (S1P) 是 S1P1-5 受体 (S1P1-5 receptors) 的激动剂和 GPR3、GPR6、GPR12 的配体。Sphingosine-1-phosphate 是细胞内的第二信使,动员 Ca2+ 作为 G 蛋白偶联受体的细胞外配体。Sphingosine-1-phosphate 是由鞘磷脂 (HY-113498) 或其他膜磷脂生成的重要脂质介质。

天然产物

Sphingosine-1-phosphate
Cat.No: T21500
Synonym: S1P
Target: Endogenous Metabolite, S1P Receptor, LPL Receptor
TargetMol Loading
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