Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3617 |
Ivosidenib
艾伏尼布,AG-120 |
Dehydrogenase; Isocitrate Dehydrogenase (IDH) | Metabolism |
Ivosidenib (AG-120) 是一种口服具有活力的异柠檬酸脱氢酶 1 的突变体酶 (mIDH1 enzyme) 抑制剂,能够使 d-2- hydroxyglutatrate (2-HG) 在体内降低。它具有良好的的安全性和临床活性,具有研究 AML 的潜力。 | |||
T13438 |
(R,S)-Ivosidenib
(R,S)-AG-120 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib . | |||
T22253 |
AG-120 (racemic)
1-(4-氰基-2-吡啶基)-5-氧代-L-脯氨酰-2-(2-氯苯基)-N-(3,3-二氟环丁基)-N2-(5-氟-3-吡啶基)甘氨酰胺 |
Dehydrogenase | Metabolism |
AG-120 (racemic) 是 AG-120 的外消旋混合物,是一种可口服的异柠檬酸脱氢酶 1 型 (IDH1) 抑制剂,具有潜在的抗肿瘤活性。 |