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Cat. No. Product Name Target Signaling Pathways
T70758 Copanlisib HCl hydrate

Copanlisib Dihydrochloride is a novel phosphoinositide 3-kinase (pi3k) inhibitor, inhibiting the activation of the pi3k signaling pathway, resulting in inhibition of tumor cell growth and survival in susceptible tumor cell populations
T14998 Copanlisib dihydrochloride

库潘尼西盐酸,BAY 80-6946 dihydrochloride

Apoptosis; PI3K; mTOR Apoptosis; PI3K/Akt/mTOR signaling
Copanlisib dihydrochloride (BAY 80-6946 dihydrochloride) 是一种选择性和 ATP 竞争性的泛 I 类 PI3K 抑制剂。它具有优越的抗肿瘤活性,对除 mTOR 以外的其他脂质和蛋白激酶的选择性也超过 2,000 倍。
T6322 Copanlisib

BAY 80-6946,可泮利塞,库潘尼西

Apoptosis; PI3K Apoptosis; PI3K/Akt/mTOR signaling
Copanlisib (BAY 80-6946) 是一种选择性的和 ATP 竞争性的泛 I 类PI3K 抑制剂,具有抗肿瘤活性,对PI3Kα,PI3Kδ,PI3Kβ和PI3Kγ的IC50分别为 0.5 nM、0.7 nM、3.7 nM 和 6.4 nM。

化合物

Copanlisib HCl hydrate
Cat.No: T70758
Synonym:
Target:
Copanlisib dihydrochloride
Cat.No: T14998
Synonym: 库潘尼西盐酸,BAY 80-6946 dihydrochloride
Target: Apoptosis, PI3K, mTOR
Copanlisib
Cat.No: T6322
Synonym: BAY 80-6946,可泮利塞,库潘尼西
Target: Apoptosis, PI3K
TargetMol Loading
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