4
1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1021 |
(R)-Lansoprazole
Dexlansoprazole,右旋兰索拉唑,T 168390,TAK 390,R-(+)-Lansoprazole |
Proton pump | Membrane transporter/Ion channel |
(R)-Lansoprazole (T 168390) 是Lansoprazole 的R 型异构体。Lansoprazole 是口服有效的质子泵抑制剂,能抑制胃酸生成。Lansoprazole 是中性鞘磷脂酶(N-SMase)的抑制剂(外泌体抑制剂),能透过血脑屏障。 | |||
T20714 |
Levolansoprazole
左旋兰索拉唑,(S)-Lansoprazole,(-)-Lansoprazole |
Proton pump | Membrane transporter/Ion channel |
Levolansoprazole ((S)-Lansoprazole) 是一种质子泵抑制剂,不可逆地抑制壁细胞中 H+/K+ 刺激的 ATPase 泵 (IC50: 5.2 µM)。它还抑制分离的犬壁细胞中的酸形成(IC50:82 µM)。 (R)-和 (S)-兰索拉唑均具有药理活性,具有相似的效力。 | |||
T11816 |
Lansoprazole-d4
AG-1749 D4,Lansoprazole D4 |
Proton pump | Membrane transporter/Ion channel |
Lansoprazole D4 (AG-1749 D4) is a deuterium labeled Lansoprazole. Lansoprazole is an inhibitor of proton pump which prevents the stomach from producing acid. | |||
T0674 |
Lansoprazole
兰索拉唑,A-65006,AG-1749 |
Proton pump; Phospholipase; Antibacterial | Membrane transporter/Ion channel; Metabolism; Microbiology/Virology |
Lansoprazole (A-65006) 是一种可抑制胃酸生成的质子泵抑制剂。它是中性鞘磷脂酶的外泌体抑制剂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T21651 |
Lansoprazole sodium
兰索拉唑钠,Lansoprazole (sodium), AG-1749 sodium |
Proton pump; Phospholipase; Antibacterial | Membrane transporter/Ion channel; Metabolism; Microbiology/Virology |
Lansoprazole sodium (Lansoprazole (sodium)) 是一种质子泵抑制剂,是中性鞘磷脂酶的外泌体抑制剂,能抑制胃酸生成。 |