Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T67739 |
BMY-14802
alpha-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazine butanol |
Sigma receptor | GPCR/G Protein |
BMY-14802 (alpha-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazine butanol)是一种选择性的、口服活性的sigma-1拮抗剂,IC50为112nM。 | |||
T22612 |
BMY-14802 hydrochloride
BMS 181100 hydrochloride,BMY-14802-1,BMY 14802 hydrochloride |
Sigma receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
BMY-14802 hydrochloride (BMS 181100 hydrochloride) 是一种选择性的 σ 受体拮抗剂 (IC50 = 112 nM),具有抗精神病作用。 BMY-14802 hydrochloride 是 α1-肾上腺素能受体和 5-HT1A 的激动剂。 |