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Cat. No. Product Name Target Signaling Pathways
T8214 Kushenol E

苦参醇E,Flemiphilippinin D

IDO; Indoleamine 2,3-Dioxygenase (IDO) Metabolism
Kushenol E (Flemiphilippinin D) 是一种分离自Sophora flavescens 中的类黄酮,是一种IDO1的非竞争性抑制剂,其IC50=7.7 µM,Ki=为 9.5 µM,具有抗肿瘤特性。
TN1841 Kushenol A

苦参新醇 A,Leachianone E

cAMP GPCR/G Protein
Kushenol A is a kind of Adenosine 3', 5'-cyclic monophosphate(cAMP)phosphodiesterase inhibitiors, it shows selective alpha-glucosidase inhibitory activity. Kushenol A and kushenol C exhibit inhibitory activity against Sodium-dependent glucose cotransporter 2(SGLT2).

天然产物

Kushenol E
Cat.No: T8214
Synonym: 苦参醇E,Flemiphilippinin D
Target: IDO, Indoleamine 2,3-Dioxygenase (IDO)
Kushenol A
Cat.No: TN1841
Synonym: 苦参新醇 A,Leachianone E
Target: cAMP
TargetMol Loading
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