Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1159 |
Leflunomide
SU101,RS-34821,HWA486,来氟米特 |
Others; Dehydrogenase; AhR | Immunology/Inflammation; Metabolism; Others |
Leflunomide (HWA486) 是嘧啶合成抑制剂,能够抑制二氢乳清酸脱氢酶,具有抗风湿的活性。 | |||
T11020 |
DHODH-IN-11
|
Dehydrogenase; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism |
DHODH-IN-11 是一种来氟米特衍生物和弱二氢乳清酸脱氢酶 (DHODH) 抑制剂,pKa 为 5.03 | |||
T7534 |
Teriflunomide
A 77-1726,特立氟胺 |
Others | Others |
Teriflunomide (A 77-1726) 是一种来氟米特的活性代谢产物,能够抑制嘧啶合成,有效降低T 细胞和B 细胞增殖,可用于研究类风湿性关节炎。 |