Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2588 |
Ivacaftor
Ivacaftor (VX-770),VX-770,依伐卡托 |
CFTR; Autophagy | Autophagy; Membrane transporter/Ion channel |
Ivacaftor (VX-770) 是一种 CFTR 增强剂,靶向G551D-CFTR 和F508del-CFTR 的EC50分别为100 和 25 nM。 | |||
T27098 |
Ivacaftor-D9
deutivacaftor,CTP-656 |
||
CTP-656, a cystic fibrosis transmembrane conductance regulator (CFTR) channel activator, is used potentially for the treatment of cystic fibrosis. | |||
T13742L |
Ivacaftor hydrate
VX-770 hydrate |
Others | Others |
Ivacaftor hydrate is an orally bioavailable CFTR potentiator. It also is used for cystic fibrosis treatment. | |||
T13742 |
Ivacaftor benzenesulfonate
VX-770 benzenesulfonate |
Others | Others |
Ivacaftor benzenesulfonate used for cystic fibrosis treatment. is an orally bioavailable CFTR potentiator. |