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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T60123 |
Chimmitecan
(S)-9-Allyl-10-hydroxycamptothecin,吉米替康 |
Topoisomerase | DNA Damage/DNA Repair |
Chimmitecan ((S)-9-Allyl-10-hydroxycamptothecin) 是一种topoisomerase I 抑制剂,在体内、外表现有效的活性。 | |||
T67812 |
Tenifatecan
SN2310 |
||
Tenifatecan (SN2310) 是一种高度亲脂性的7-乙基-10-羟基喜树碱(SN)制剂,具有潜在的抗肿瘤活性。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1521 |
(±)-10-Hydroxycamptothecin
Hydroxy Camptothecine,10-羟基喜树碱,10-Hydroxycamptothecin |
Topoisomerase | DNA Damage/DNA Repair |
(±)-10-Hydroxycamptothecin (Hydroxy Camptothecine) 是一种从喜树茎木中分离出来的生物碱,抑制拓扑异构酶 I 活性,具有广谱抗肿瘤活性。 | |||
T2764 |
(S)-10-Hydroxycamptothecin
10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT |
Apoptosis; Topoisomerase | Apoptosis; DNA Damage/DNA Repair |
(S)-10-Hydroxycamptothecin (10-HCPT) 是一种从喜树中分离的 DNA 拓扑异构酶 I 抑制剂。它显著诱导细胞凋亡,可研究肝癌、胃癌、结肠癌和白血病。 | |||
T4952 |
9-Hydroxycamptothecin
9-HCPT,9-羟基喜树碱,10-Hydroxycampothecin |
Topoisomerase | DNA Damage/DNA Repair |
9-Hydroxycampothecin 是具有抗癌活性的喜树碱衍生物。 | |||
TN2460 |
12-Ethyl-9-hydroxycamptothecin
7-乙基-10-羟基喜树碱,7-Ethyl-10-Hydroxy-Camptothecin |
Others | Others |
12-Ethyl-9-hydroxycamptothecin 是一种 Camptothecin 的衍生物。其中Camptothecin (CPT) 是一种生物碱,也是 DNA 拓扑异构酶I 抑制剂(IC50:679 nM)。 |