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E1/E2/E3 Enzyme inhibitor kit

Catalog No. CL0137

E1/E2/E3 Enzyme inhibitor kit 包含 E1/E2/E3泛素化酶抑制剂,泛素化是指泛素在一系列酶的催化作用下共价结合到靶蛋白上的过程,包括 E1泛素激活酶、E2泛素偶联酶 和 E3泛素连接酶。泛素化调控蛋白质稳定性、亚细胞定位、活性以及相互作用等方面,参与免疫反应调控、线粒体自噬DNA 损伤修复、细胞周期调控、表观遗传调控、细胞凋亡和蛋白质降解等生理过程。TargetMol 为您提供50种精选 E1/E2/E3泛素化酶抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
E1/E2/E3 Enzyme inhibitor kit
规格 价格/CNY 货期 数量
10 μL * 10 mM (in DMSO) ¥ 1,500 4-6周
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产品组成

IDCompoundCASMWConcentrationTarget
T1493BH3I-1300817-68-9400.3110mMBcl; E1/E2/E3 Enzyme; MDM-2/p53
T2158Nutlin-3548472-68-0581.4910mME1/E2/E3 Enzyme; MDM-2/p53
T2243Serdemetan881202-45-5328.4210mMApoptosis; E1/E2/E3 Enzyme; MDM-2/p53; Mdm2; p53
T2947Indole-3-carbinol700-06-1147.1710mMAryl Hydrocarbon Receptor; E1/E2/E3 Enzyme; Endogenous Metabolite; NF-κB; p53
T3110PRT416531083-55-3235.2410mMBMI-1; E1/E2/E3 Enzyme
T3317SZL P1-41222716-34-9420.5210mMApoptosis; E1/E2/E3 Enzyme
T3517RO89941309684-94-3613.5110mME1/E2/E3 Enzyme; MDM-2/p53; Mdm2; p53
T3653MX691005264-47-0474.5710mME1/E2/E3 Enzyme; IAP; MDM-2/p53; Mdm2
T4036Solasodine126-17-0413.6510mMAntifungal; Apoptosis; E1/E2/E3 Enzyme; MDM-2/p53
T4253Skp2 Inhibitor C1432001-69-9465.3410mME1/E2/E3 Enzyme
T6023Nutlin-3a675576-98-4581.4910mMApoptosis; Autophagy; E1/E2/E3 Enzyme; MDM-2/p53
T6149YH239-EE1364488-67-4504.4110mMApoptosis; E1/E2/E3 Enzyme; MDM-2/p53
T6254Idasanutlin1229705-06-9616.4810mME1/E2/E3 Enzyme; MDM-2/p53; Mdm2
T6332Pevonedistat905579-51-3443.5210mME1/E2/E3 Enzyme; NEDD8
T6614Nutlin-3b675576-97-3581.4910mME1/E2/E3 Enzyme; MDM-2/p53; Mdm2
T6629PYR-41418805-02-4371.310mMApoptosis; E1/E2/E3 Enzyme
T6965RG7112939981-39-2727.7810mME1/E2/E3 Enzyme; MDM-2/p53; Mdm2
T6611NSC697923343351-67-7267.2610mMApoptosis; E1/E2/E3 Enzyme
T6S2123Ginkgolic Acid22910-60-7346.5110mME1/E2/E3 Enzyme
T5199COH0001534358-79-6419.4710mME1/E2/E3 Enzyme
T73792-D08144707-18-6270.2410mME1/E2/E3 Enzyme; TAM Receptor
T7415DKM 2-9365836-72-8243.6910mME1/E2/E3 Enzyme
T7889C25-1401358099-18-9457.610mME1/E2/E3 Enzyme; NF-κB; TNF
T11980MD-2242136247-12-4889.810mME1/E2/E3 Enzyme; MDM-2/p53; Mdm2; PROTACs
T8564BC-13821013753-99-5459.5610mME1/E2/E3 Enzyme
T10703Mezigdomide2259648-80-9567.6110mMApoptosis; E1/E2/E3 Enzyme; Molecular Glues
T16974TAK-2431450833-55-2519.5210mMApoptosis; E1/E2/E3 Enzyme; NF-κB
T8816NAE-IN-M22864420-54-2363.3210mMApoptosis; E1/E2/E3 Enzyme
T4S0181Hinokiflavone19202-36-9538.510mMBCL; E1/E2/E3 Enzyme; MMP
T13349WS-3832247544-02-9498.4610mME1/E2/E3 Enzyme
T16888SJ-172550431979-47-4428.8710mME1/E2/E3 Enzyme; MDM-2/p53; Mdm2
T8929BC16182222094-18-8415.4510mMAMPK; E1/E2/E3 Enzyme; Mitophagy
TQ0231NVP-CGM0971313363-54-0659.2610mME1/E2/E3 Enzyme; MDM-2/p53; Mdm2
T8428Subasumstat1858276-04-6578.110mME1/E2/E3 Enzyme
T5555Siremadlin1448867-41-1555.4110mME1/E2/E3 Enzyme; MDM-2/p53
TQ0127Navtemadlin1352066-68-2568.5510mME1/E2/E3 Enzyme; MDM-2/p53; Mdm2
T25465GS143916232-21-8466.4610mME1/E2/E3 Enzyme; IκB/IKK; NF-κB
T9236WSB1 Degrader 12306039-66-5334.4110mME1/E2/E3 Enzyme
T12261NSC2320031905453-18-0169.1410mME1/E2/E3 Enzyme
T13090TAS4464 hydrochloride1848959-11-4542.9710mME1/E2/E3 Enzyme; NEDD8
T16102ML-7921644342-14-2551.4110mME1/E2/E3 Enzyme
T16901SMIP004143360-00-3205.310mME1/E2/E3 Enzyme;Apoptosis
T24136Heclin890605-54-6283.3210mME1/E2/E3 Enzyme
T16699PYZD-4409423148-78-1351.6710mME1/E2/E3 Enzyme
T13412ZM2232031177-48-5502.5310mME1/E2/E3 Enzyme
T3798Ziyuglycoside I35286-58-9766.9710mMApoptosis; MDM-2/p53
T21773SP-1411253491-42-7324.3810mMMDM-2/p53; Mdm2
T21578NSC 668116964-62-1340.4210mMMDM-2/p53
T28509RDR03871286008-51-3408.8110mMMdm2
T14303Alrizomadlin1818393-16-6642.5910mMMdm2

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产品应用

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包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输
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