E1/E2/E3 Enzyme inhibitor kit 包含 E1/E2/E3泛素化酶抑制剂,泛素化是指泛素在一系列酶的催化作用下共价结合到靶蛋白上的过程,包括 E1泛素激活酶、E2泛素偶联酶 和 E3泛素连接酶。泛素化调控蛋白质稳定性、亚细胞定位、活性以及相互作用等方面,参与免疫反应调控、线粒体自噬、DNA 损伤修复、细胞周期调控、表观遗传调控、细胞凋亡和蛋白质降解等生理过程。TargetMol 为您提供50种精选 E1/E2/E3泛素化酶抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1493 | BH3I-1 | 300817-68-9 | 400.31 | 10mM | Bcl; E1/E2/E3 Enzyme; MDM-2/p53 |
T2158 | Nutlin-3 | 548472-68-0 | 581.49 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53 |
T2243 | Serdemetan | 881202-45-5 | 328.42 | 10mM | Apoptosis; E1/E2/E3 Enzyme; MDM-2/p53; Mdm2; p53 |
T2947 | Indole-3-carbinol | 700-06-1 | 147.17 | 10mM | Aryl Hydrocarbon Receptor; E1/E2/E3 Enzyme; Endogenous Metabolite; NF-κB; p53 |
T3110 | PRT4165 | 31083-55-3 | 235.24 | 10mM | BMI-1; E1/E2/E3 Enzyme |
T3317 | SZL P1-41 | 222716-34-9 | 420.52 | 10mM | Apoptosis; E1/E2/E3 Enzyme |
T3517 | RO8994 | 1309684-94-3 | 613.51 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2; p53 |
T3653 | MX69 | 1005264-47-0 | 474.57 | 10mM | E1/E2/E3 Enzyme; IAP; MDM-2/p53; Mdm2 |
T4036 | Solasodine | 126-17-0 | 413.65 | 10mM | Antifungal; Apoptosis; E1/E2/E3 Enzyme; MDM-2/p53 |
T4253 | Skp2 Inhibitor C1 | 432001-69-9 | 465.34 | 10mM | E1/E2/E3 Enzyme |
T6023 | Nutlin-3a | 675576-98-4 | 581.49 | 10mM | Apoptosis; Autophagy; E1/E2/E3 Enzyme; MDM-2/p53 |
T6149 | YH239-EE | 1364488-67-4 | 504.41 | 10mM | Apoptosis; E1/E2/E3 Enzyme; MDM-2/p53 |
T6254 | Idasanutlin | 1229705-06-9 | 616.48 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T6332 | Pevonedistat | 905579-51-3 | 443.52 | 10mM | E1/E2/E3 Enzyme; NEDD8 |
T6614 | Nutlin-3b | 675576-97-3 | 581.49 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T6629 | PYR-41 | 418805-02-4 | 371.3 | 10mM | Apoptosis; E1/E2/E3 Enzyme |
T6965 | RG7112 | 939981-39-2 | 727.78 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T6611 | NSC697923 | 343351-67-7 | 267.26 | 10mM | Apoptosis; E1/E2/E3 Enzyme |
T6S2123 | Ginkgolic Acid | 22910-60-7 | 346.51 | 10mM | E1/E2/E3 Enzyme |
T5199 | COH000 | 1534358-79-6 | 419.47 | 10mM | E1/E2/E3 Enzyme |
T7379 | 2-D08 | 144707-18-6 | 270.24 | 10mM | E1/E2/E3 Enzyme; TAM Receptor |
T7415 | DKM 2-93 | 65836-72-8 | 243.69 | 10mM | E1/E2/E3 Enzyme |
T7889 | C25-140 | 1358099-18-9 | 457.6 | 10mM | E1/E2/E3 Enzyme; NF-κB; TNF |
T11980 | MD-224 | 2136247-12-4 | 889.8 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2; PROTACs |
T8564 | BC-1382 | 1013753-99-5 | 459.56 | 10mM | E1/E2/E3 Enzyme |
T10703 | Mezigdomide | 2259648-80-9 | 567.61 | 10mM | Apoptosis; E1/E2/E3 Enzyme; Molecular Glues |
T16974 | TAK-243 | 1450833-55-2 | 519.52 | 10mM | Apoptosis; E1/E2/E3 Enzyme; NF-κB |
T8816 | NAE-IN-M22 | 864420-54-2 | 363.32 | 10mM | Apoptosis; E1/E2/E3 Enzyme |
T4S0181 | Hinokiflavone | 19202-36-9 | 538.5 | 10mM | BCL; E1/E2/E3 Enzyme; MMP |
T13349 | WS-383 | 2247544-02-9 | 498.46 | 10mM | E1/E2/E3 Enzyme |
T16888 | SJ-172550 | 431979-47-4 | 428.87 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T8929 | BC1618 | 2222094-18-8 | 415.45 | 10mM | AMPK; E1/E2/E3 Enzyme; Mitophagy |
TQ0231 | NVP-CGM097 | 1313363-54-0 | 659.26 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T8428 | Subasumstat | 1858276-04-6 | 578.1 | 10mM | E1/E2/E3 Enzyme |
T5555 | Siremadlin | 1448867-41-1 | 555.41 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53 |
TQ0127 | Navtemadlin | 1352066-68-2 | 568.55 | 10mM | E1/E2/E3 Enzyme; MDM-2/p53; Mdm2 |
T25465 | GS143 | 916232-21-8 | 466.46 | 10mM | E1/E2/E3 Enzyme; IκB/IKK; NF-κB |
T9236 | WSB1 Degrader 1 | 2306039-66-5 | 334.41 | 10mM | E1/E2/E3 Enzyme |
T12261 | NSC232003 | 1905453-18-0 | 169.14 | 10mM | E1/E2/E3 Enzyme |
T13090 | TAS4464 hydrochloride | 1848959-11-4 | 542.97 | 10mM | E1/E2/E3 Enzyme; NEDD8 |
T16102 | ML-792 | 1644342-14-2 | 551.41 | 10mM | E1/E2/E3 Enzyme |
T16901 | SMIP004 | 143360-00-3 | 205.3 | 10mM | E1/E2/E3 Enzyme;Apoptosis |
T24136 | Heclin | 890605-54-6 | 283.32 | 10mM | E1/E2/E3 Enzyme |
T16699 | PYZD-4409 | 423148-78-1 | 351.67 | 10mM | E1/E2/E3 Enzyme |
T13412 | ZM223 | 2031177-48-5 | 502.53 | 10mM | E1/E2/E3 Enzyme |
T3798 | Ziyuglycoside I | 35286-58-9 | 766.97 | 10mM | Apoptosis; MDM-2/p53 |
T21773 | SP-141 | 1253491-42-7 | 324.38 | 10mM | MDM-2/p53; Mdm2 |
T21578 | NSC 66811 | 6964-62-1 | 340.42 | 10mM | MDM-2/p53 |
T28509 | RDR03871 | 286008-51-3 | 408.81 | 10mM | Mdm2 |
T14303 | Alrizomadlin | 1818393-16-6 | 642.59 | 10mM | Mdm2 |