Casein Kinase inhibitor kit 包含酪蛋白激酶抑制剂,酪蛋白激酶催化肽链中邻近酸性氨基酸残基的丝氨酸/苏氨酸磷酸化的酶,主要包括酪蛋白激酶1和酪蛋白激酶2,在细胞分裂与凋亡、DNA 修复、P53调控、周期性节律等多种机体生理活动中发挥重要作用。TargetMol 为您提供32种精选酪蛋白激酶抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0465 | Ellagic acid | 476-66-4 | 302.19 | 10mM | Carbonic Anhydrase; Casein Kinase; Endogenous Metabolite; Hedgehog/Smoothened; PKA; PKC; Reactive Oxygen Species; Syk; Topoisomerase |
T1828 | TTP 22 | 329907-28-0 | 330.42 | 10mM | Casein Kinase |
T1877 | LH846 | 639052-78-1 | 316.81 | 10mM | Casein Kinase |
T2008 | LY294002 | 154447-36-6 | 307.34 | 10mM | Apoptosis; Autophagy; Casein Kinase; DNA-PK; PI3K |
T2048 | LY-364947 | 396129-53-6 | 272.3 | 10mM | Casein Kinase; MLK; RIP kinase; TGF-beta/Smad |
T2259 | Silmitasertib | 1009820-21-6 | 349.77 | 10mM | Autophagy; Casein Kinase |
T2440 | IC261 | 186611-52-9 | 311.33 | 10mM | Apoptosis; Casein Kinase; CDK |
T2449 | D4476 | 301836-43-1 | 398.41 | 10mM | ALK; Apoptosis; Autophagy; Casein Kinase |
T2695 | TBB | 17374-26-4 | 434.71 | 10mM | Casein Kinase; CDK; GSK-3 |
T2702 | IWP-2 | 686770-61-6 | 466.6 | 10mM | Casein Kinase; Porcupine; Wnt/beta-catenin |
T2869 | Emodin | 518-82-1 | 270.24 | 10mM | Autophagy; Casein Kinase; SARS-CoV |
T3073 | PF-670462 | 950912-80-8 | 410.32 | 10mM | Casein Kinase |
T3972 | SR-3029 | 1454585-06-8 | 480.45 | 10mM | Casein Kinase |
T6150 | TAK-715 | 303162-79-0 | 399.51 | 10mM | Casein Kinase; JNK; p38 MAPK |
T6735 | XL413 hydrochloride | 1169562-71-3 | 326.18 | 10mM | Casein Kinase; CDK; Pim |
T4645 | TA-01 | 1784751-18-3 | 351.32 | 10mM | Autophagy; Casein Kinase; p38 MAPK |
T5056 | PF-4800567 | 1188296-52-7 | 359.8 | 10mM | Casein Kinase |
T5358 | Longdaysin | 1353867-91-0 | 335.33 | 10mM | Casein Kinase; CDK; ERK |
T5393 | CK1-IN-1 | 1784751-20-7 | 383.39 | 10mM | Casein Kinase; p38 MAPK |
T7390 | DMAT | 749234-11-5 | 476.79 | 10mM | Casein Kinase |
T15024 | Silmitasertib sodium salt | 1309357-15-0 | 371.75 | 10mM | Autophagy; Casein Kinase |
T14069 | A-3 hydrochloride | 78957-85-4 | 321.22 | 10mM | CaMK; Casein Kinase; PKA; PKC |
T8987 | Epiblastin A | 16470-02-3 | 287.71 | 10mM | Casein Kinase |
T7949 | NCC007 | 2342583-66-6 | 447.5 | 10mM | Casein Kinase |
T9356 | (E/Z)-GO289 | 694522-87-7 | 419.3 | 10mM | Casein Kinase |
T19913 | CKI-7 | 1177141-67-1 | 358.67 | 10mM | Casein Kinase; CDK; ROCK; S6 Kinase; SGK |
T35557 | CK2 inhibitor 2 | 2641079-92-5 | 392.84 | 10mM | Casein Kinase |
T60005 | WAY-296817 | 349438-74-0 | 328.39 | 10mM | Casein Kinase |
T10547 | BioE-1115 | 1268863-35-9 | 339.36 | 10mM | Casein Kinase;Serine/threonin kinase |
T21915 | TBCA | 934358-00-6 | 463.74 | 10mM | Casein Kinase |
T10827 | CK2/ERK8-IN-1 | 1085822-09-8 | 534.82 | 10mM | Casein Kinase;ERK;Pim;DYRK;Apoptosis |
T60067 | WAY-297174 | 442571-27-9 | 268.36 | 10mM | Casein Kinase |