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9

抑制剂 & 化合物

1

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Cat. No. Product Name Target Signaling Pathways
T19480 NO-prednisolone

NCX-1015

IL Receptor Immunology/Inflammation
NO-prednisolone (NCX-1015) 是一种有效刺激体内IL-10产生的化合物,是一种释放一氧化氮(NO)的Prednisolone 衍生物。
T0208 Prednisolone disodium phosphate

泼尼松龙21-磷酸二钠,Prednisolone phosphate sodium,Prednisolone 21-phosphate disodium,泼尼松龙磷酸钠

Glucocorticoid Receptor Endocrinology/Hormones
Prednisolone disodium phosphate是一种合成的糖皮质素,具有抗炎和免疫调节作用。
T0337 Prednisolone acetate

Omnipred,醋酸泼尼松龙,Prednisolone-21-acetate

Glucocorticoid Receptor Endocrinology/Hormones
Prednisolone acetate (Omnipred) 是一种肾上腺皮质激素类药物,具有抗炎、抗过敏和抑制免疫等多种药理活性。
T8339 16α-Hydroxyprednisolone

16alpha-羟基泼尼松龙,16alpha-Hydroxyprednisolone

Others; Drug Metabolite Metabolism; Others
16α-Hydroxyprednisolone 是糖皮质激素布地奈德 22(R) epimer 构型的代谢物,经过 CYP3A 酶代谢生成。
T22367 Methylprednisolone succinate

Methylprednisolone hemisuccinate,Methylprednisolone hydrogen succinate,甲基泼尼松龙琥珀酸酯

Glucocorticoid Receptor Endocrinology/Hormones
Methylprednisolone succinate (Methylprednisolone hemisuccinate) 是合成的糖皮质激素,常用作抗炎剂。
T12507 Prednisolone farnesylate

泼尼松龙法尼酯,PNF21

Others Others
Prednisolone farnesylate is a novel transdermal corticosteroid with anti-inflammatory activity.
T13825 Prednisolone hemisuccinate

泼尼松龙半琥珀酸酯,Prednisolone 21-hemisuccinate

Others Others
Prednisolone hemisuccinate is a synthetic glucocorticoid, and is treatment a variety of inflammatory and auto-immune conditions.
T21338 Methylprednisolone Acetate

Depo-Medrate,Depometicort,Depo-Medrin,Depo-medrol,Depomedrone,Lemod

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Methylprednisolone Acetate(Depo-Medrate) 具有抑制氧自由基的能力,可用于治疗急性脊髓损伤。
T29328 21-deacetyldeflazacort

Others Others
21-deacetyldeflazacort 是 Deflazacort 的代谢物,它是一种全身性皮质类固醇和泼尼松龙的衍生物。

化合物

NO-prednisolone
Cat.No: T19480
Synonym: NCX-1015
Target: IL Receptor
Prednisolone disodium phosphate
Cat.No: T0208
Synonym: 泼尼松龙21-磷酸二钠,Prednisolone phosphate sodium,Prednisolone 21-phosphate disodium,泼尼松龙磷酸钠
Target: Glucocorticoid Receptor
Prednisolone acetate
Cat.No: T0337
Synonym: Omnipred,醋酸泼尼松龙,Prednisolone-21-acetate
Target: Glucocorticoid Receptor
16α-Hydroxyprednisolone
Cat.No: T8339
Synonym: 16alpha-羟基泼尼松龙,16alpha-Hydroxyprednisolone
Target: Others, Drug Metabolite
Methylprednisolone succinate
Cat.No: T22367
Synonym: Methylprednisolone hemisuccinate,Methylprednisolone hydrogen succinate,甲基泼尼松龙琥珀酸酯
Target: Glucocorticoid Receptor
Prednisolone farnesylate
Cat.No: T12507
Synonym: 泼尼松龙法尼酯,PNF21
Target: Others
Prednisolone hemisuccinate
Cat.No: T13825
Synonym: 泼尼松龙半琥珀酸酯,Prednisolone 21-hemisuccinate
Target: Others
Methylprednisolone Acetate
Cat.No: T21338
Synonym: Depo-Medrate,Depometicort,Depo-Medrin,Depo-medrol,Depomedrone,Lemod
Target: Reactive Oxygen Species
21-deacetyldeflazacort
Cat.No: T29328
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1560 Prednisolone

氢化泼尼松,Predonine,Hydroretrocortine,泼尼松龙,Metacortandralone

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Prednisolone (Hydroretrocortine) 是有口服活性的皮质类固醇和糖皮质激素。它的抗炎特性约为氢化可的松的四倍,同时减少了水和盐的保留。它能够用于眼部抗炎研究。

天然产物

Prednisolone
Cat.No: T1560
Synonym: 氢化泼尼松,Predonine,Hydroretrocortine,泼尼松龙,Metacortandralone
Target: Glucocorticoid Receptor, Endogenous Metabolite
TargetMol Loading
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