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抑制剂 & 化合物

1

天然产物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T71611 αSyn-IN-576755

αSyn-IN-576755 is a novel inhibitor of αSyn fibrillization, blocking fibril growth and suppressing A53T αSyn neurotoxicity.
T61787 SYN20028567

SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].
T83726 Tat-βsyn-degron TFA

Tat-βsyn-degron是一种降低α-synuclein表达的肽。其结构包括HIV-1 Tat质膜跨导域、与β-synuclein氨基酸36-45相对应的α-synuclein结合域βsyn,以及蛋白酶体定向域degron。Tat-βsyn-degron能够与重组α-synuclein结合,并在大鼠初级皮质神经元培养中降低α-synuclein水平。
T83875 HUP-55

HUP-55是一种脯氨酸内肽酶的抑制剂(IC50 = 5 nM)。在10 µM的浓度下,它可减少Neuro2a细胞中α-突触核蛋白二聚体的形成,促使HEK293细胞发生自噬,并降低SH-SY5Y细胞中由过氧化氢诱导的反应性氧种(ROS)产量的增加。此外,HUP-55(10 mg/kg)在通过腺病毒递送α-突触核蛋白编码载体(AAV-αSyn)诱导的帕金森病小鼠模型中,能减少患侧爪的使用和纹状体中寡聚体α-突触核蛋白水平。

化合物

αSyn-IN-576755
Cat.No: T71611
Synonym:
Target:
SYN20028567
Cat.No: T61787
Synonym:
Target:
Tat-βsyn-degron TFA
Cat.No: T83726
Synonym:
Target:
HUP-55
Cat.No: T83875
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T7846 Aegeline

Others; Antifungal Microbiology/Virology; Others
Aegeline 是从 Aegle marmelos 的叶子中分离出来的一种生物碱酰胺,有抗高血糖和抗血脂异常的活性。

天然产物

Aegeline
Cat.No: T7846
Synonym:
Target: Others, Antifungal
Cat. No. Product Name Species Expression System
TMPY-06460 Alpha-Synuclein Protein, Mouse, Recombinant (His)

alphaSYN,synuclein, α (non A4 component of amyloid precursor...

Mouse E. coli
Alpha-Synuclein Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 15.31 kDa and the accession number is O55042-1.

重组蛋白

Alpha-Synuclein Protein, Mouse, Recombinant (His)
Cat.No: TMPY-06460
Species: Mouse
Expression System: E. coli
TargetMol Loading
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