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Cat. No. | Product Name | Target | Signaling Pathways |
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T71611 | αSyn-IN-576755 | ||
αSyn-IN-576755 is a novel inhibitor of αSyn fibrillization, blocking fibril growth and suppressing A53T αSyn neurotoxicity. | |||
T61787 |
SYN20028567
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SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1]. | |||
T83726 |
Tat-βsyn-degron TFA
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Tat-βsyn-degron是一种降低α-synuclein表达的肽。其结构包括HIV-1 Tat质膜跨导域、与β-synuclein氨基酸36-45相对应的α-synuclein结合域βsyn,以及蛋白酶体定向域degron。Tat-βsyn-degron能够与重组α-synuclein结合,并在大鼠初级皮质神经元培养中降低α-synuclein水平。 | |||
T83875 |
HUP-55
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HUP-55是一种脯氨酸内肽酶的抑制剂(IC50 = 5 nM)。在10 µM的浓度下,它可减少Neuro2a细胞中α-突触核蛋白二聚体的形成,促使HEK293细胞发生自噬,并降低SH-SY5Y细胞中由过氧化氢诱导的反应性氧种(ROS)产量的增加。此外,HUP-55(10 mg/kg)在通过腺病毒递送α-突触核蛋白编码载体(AAV-αSyn)诱导的帕金森病小鼠模型中,能减少患侧爪的使用和纹状体中寡聚体α-突触核蛋白水平。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T7846 |
Aegeline
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Others; Antifungal | Microbiology/Virology; Others |
Aegeline 是从 Aegle marmelos 的叶子中分离出来的一种生物碱酰胺,有抗高血糖和抗血脂异常的活性。 |
Cat. No. | Product Name | Species | Expression System |
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TMPY-06460 |
Alpha-Synuclein Protein, Mouse, Recombinant (His)
alphaSYN,synuclein, α (non A4 component of amyloid precursor... |
Mouse | E. coli |
Alpha-Synuclein Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 15.31 kDa and the accession number is O55042-1. |