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Cat. No. Product Name Target Signaling Pathways
T6086 Clopamide

Brinaldix,Adurix,Aquex,氯帕胺

Sodium Channel Membrane transporter/Ion channel
Clopamide (Brinaldix) 是口服有效的噻嗪类利尿剂,对钠耦合的氯离子共转运蛋白 SLC12A3有抑制作用。Clopamide 在高血压和心力衰竭中具有研究价值。
T0275 Meticrane

美替克仑,Fontiliz,Arresten,蒲硫杂茶磺胺

Chloride channel; Sodium Channel Membrane transporter/Ion channel
Meticrane (Arresten) 是一种磺胺类衍生物,具有类似噻嗪类利尿剂的活性,可于研究原发性高血压。
T31777 Fenquizone

M.G. 13054

Others Others
Fenquizone (M.G. 13054) 是一种噻嗪样利尿剂,具有慢性抗高血压作用。Fenquizone 可用于水肿和高血压的研究。
T82735 Chlorthalidone impurity

Chlorthalidoneimpurity,作为Chlorthalidone的代谢物,该物质属于噻嗪类利尿剂,主要用于高血压的研究。
T35876 Chlorthalidone Impurity G

Chlorthalidone impurity G is a potential impurity found in commercial preparations of chlorthalidone that has moderate antihypertensive effects. Chlorthalidone is a thiazide-like diuretic that inhibits the Na+/Cl- cotransporter in the distal convoluted tubule of the kidney, which prevents reabsorption of sodium and chloride leading to a reduction in plasma volume and cardiac output. It also inhibits carbonic anhydrase (CA), including the isoforms CAVB, VII, IX, XII, and XIII (Kis = 2.8-23 nM) an...

化合物

Clopamide
Cat.No: T6086
Synonym: Brinaldix,Adurix,Aquex,氯帕胺
Target: Sodium Channel
Meticrane
Cat.No: T0275
Synonym: 美替克仑,Fontiliz,Arresten,蒲硫杂茶磺胺
Target: Chloride channel, Sodium Channel
Fenquizone
Cat.No: T31777
Synonym: M.G. 13054
Target: Others
Chlorthalidone impurity
Cat.No: T82735
Synonym:
Target:
Chlorthalidone Impurity G
Cat.No: T35876
Synonym:
Target:
TargetMol Loading
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