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Cat. No.	Product Name	Target	Signaling Pathways
TP1302	Somatostatin
	Somatostatin, also known as growth hormone-inhibiting hormone, is a naturally-occurring peptide hormone of 14 or 28 amino acid residues that regulates the endocrine system. It is secreted by the D cells of the islets to inhibit the release of insulin and
TP1035L	Cyclic somatostatin Acetate(38916-34-6(free base)) Somatostatin (sheep), monoacetate (salt),Somatostatin-14,SRIF-14,monoacetate (salt)	Others	Others
	Cyclic somatostatin Acetate(38916-34-6(free base)) (Somatostatin-14) 是一种环状十四肽，可调节许多内分泌和神经系统功能。
TP2124L	Somatostatin 1-28 acetate Somatostatin 1-28 acetate(74315-46-1 Free base)	Somatostatin	GPCR/G Protein
	Somatostatin 1-28 acetate 在人源血浆中循环。血浆中约 46% 的总生长抑素样免疫反应性是由于 Somatostatin 1-28 acetate 所致。
TP1035	Cyclic somatostatin SRIF-14,合成生长抑素,环状生长激素抑制素,Somatostatin-14	Others	Others
	Cyclic somatostatin (SRIF-14) 是生长激素释放抑制因子，可用于研究胃十二指肠溃疡出血。
TP1790L	Tyr-Somatostatin-14 acetate(58100-03-1 free base)	Others	Others
	Tyr-Somatostatin-14 acetate(58100-03-1 free base) 是一种定制肽，可在 Somatostatin-14 中添加酪氨酸氨基酸。
T40680	[Tyr11]-Somatostatin [Tyr11]-Somatostatin
	[Tyr11]-Somatostatin is a neuroactive peptide utilized in proteomics research. It belongs to a class of neuroactive substances that play a role in modulating retinal physiology.
T40679	[Tyr1]-Somatostatin-14 [Tyr1]-Somatostatin-14
	[Tyr1]-Somatostatin-14 could binds to SSTR2.
T26200	Somatostatin RC 102 Somatostatin RC102,Somatostatin-RC-102,Somatostatin RC-102
	Somatostatin RC 102 is a peptide hormone. It regulates the endocrine system and affects neurotransmission and cell proliferation via interaction with G protein-coupled somatostatin receptors and inhibition of the release of numerous secondary hormones.
TP1258	Somatostatin-28 (1-12) 1-12-Somatostatin-28,Somatostatin-28 1-12
	Somatostatin-28 (1-12) is a somatostatin fragment which is monitored in brain tissue to track processing of somatostatin.
TP1823	Somatostatin-28 (1-14) Somatostatin-28 1-14
	Somatostatin-28 (1-14) is an N-terminal fragment of the neuropeptide somatostatin-28. Somatostatin 28 arises from the posttranslational cleavage of prosomatostatin, which in turn is derived from a large precursor, preprosomatostatin.
TP1810	Somatostatin-25
	Somatostatin is an endogenous neuropeptide hormone found in the brain and pancreas. Somatostatin binds several isoforms of the somatostatin receptor, exhibiting anxiolytic, antiepileptic/anticonvulsant, and anorexigenic activities.
TP2124	Somatostatin 1-28
	Somatostatin receptor agonist, derived from the post-translational cleavage of prosomatostatin.
TP1790	Tyr-Somatostatin-14
	Tyr-Somatostatin-14 is a modified peptide incorporating an additional Tyrosine (amino acid) into the structure of Somatostatin-14.
T34683	Somatostatin(3-6) Cys-lys-asn-phe
	Somatostatin(3-6) is a somatostatin fragment.
T76460	Tyr-Somatostatin-28
	Tyr-Somatostatin-28 是一种生长抑素，在 Somatostatin-28 的基础上添加了一个酪氨酸。
T2584	Octreotide SMS 201-995,奥曲肽	Somatostatin	GPCR/G Protein
	Octreotide (SMS 201-995) 是一种有效的生长激素、胰高血糖素和胰岛素抑制剂。它主要与生长抑素 2、3 和 5 亚型受体结合，可增强 Gi 活性，降低胞内 cAMP 的产生。
T83494	[D-Trp8,Tyr11] Somatostatin
	[D-Trp8,Tyr11] Somatostatin是一种somatostatin的类似物，后者是一种调节多种身体机能的激素。在该化合物中，DTrp8残基的加入可以提高其稳定性。
TP2207	Pasireotide Acetate	Somatostatin	GPCR/G Protein
	Pasireotide acetate 是长效的环己肽生长激素抑制素类似物，具有抗分泌、抗增殖和促凋亡活性。它可抑制 GH、IGF-I 和 ACTH 的分泌，可用于研究肢端肥大症和库欣病。它还可以提高生长抑素受体的激动剂活性，对sst1、2、3、4、5的pKi 分别为 8.2、9.0、9.1、小于7.0 和 9.9。
T83493	[D-Trp8] Somatostatin-14
	[D-Trp8] Somatostatin-14为一种十四肽生长抑素类似物，其活性优于天然Somatostatin。
T9692	Paltusotine	Somatostatin	GPCR/G Protein
	Paltusotine 是一种口服有效的，非肽选择性生长抑素 2 型受体激动剂。在长效生长抑素受体配体作用后，Paltusotine 仍可维持 GH 和 IGF-1 水平。
T7829	FK962	Somatostatin	GPCR/G Protein
	FK962 是抑制生长抑素释放的增强剂，具有增强认知效果。
T76461	[Nle8] Somatostatin (1-28)
	[Nle8] Somatostatin (1-28)为生长抑素(1-28)的衍生物，其特征在于第8位的甲硫氨酸被正亮氨酸所替代。该化合物能够促使淀粉酶的释放，并增加胰腺腺泡中的环AMP水平。
T83546	(D-Trp8,D-Cys14)-Somatostatin-14
	"(D-Trp8,D-Cys14)-Somatostatin-14"为一种生长抑素合成类似物，主要用于代谢相关疾病研究。
T76459	[Tyr12] Somatostatin 28 (1-14)
	[Tyr12] Somatostatin 28 (1-14)，是Somatostatin-28 (1-14)的类似物，属于神经肽生长抑素-28的N-末端片段。
T4119	Octreotide Acetate 醋酸奥曲肽,SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)	Somatostatin	GPCR/G Protein
	Octreotide Acetate (Sandostatin) 是一种长期有效的合成生长抑素八肽类似物，可抑制生长激素的分泌。
T20204	Edotreotide 依多曲肽,SMT 487,SMT487,SMT-487	Others	Others
	Edotreotide (SMT-487) 是生长抑素类似物。它与多种放射性核素联合使用，拥有研究和诊断某些类型癌症的潜能。
T76612	(D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide
	(D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide (Compound 4) 是一种生长抑素类似物，对 SSTR5、SSTR3、SSTR2、SSTR1和 SSTR4的Kd 分别为 0.61、11.05、23.5、1200 和 >1000 nM。
T80135	Tyr-(D-Dab4,Arg5,D-Trp8)-cyclo-Somatostatin-14 (4-11)
	Tyr-(D-Dab4,Arg5,D-Trp8)-cyclo-Somatostatin-14 (4-11)，一种生长抑素激动剂，用于癌症研究。
TP2045	CH 275
	Potent somatostatin receptor 1 (sst1) agonist; displays selectivity for sst1 (IC50 values are 30.9 nM, 345 nM, > 1 μM, > 10 μM and > 10μM for human sst1, sst3, sst4, sst2 and sst5 respectively). Attenuates somatostatin release in the rat nucleus accumbens
T21567L	Cyclosomatostatin Acetate Cyclosomatostatin Acetate （84211-54-1 Free base）	Somatostatin	GPCR/G Protein
	Cyclosomatostatin Acetate 是有效的生长抑素受体拮抗剂。Cyclosomatostatin Acetate 在直肠癌 (CRC) 细胞中可以抑制 SSTR1的信号传导，并降低结细胞增殖、ALDH+ 细胞群体大小和球形成。
T75842	Cyclosomatostatin TFA
	Cyclosomatostatin TFA 作为一种有效的生长抑素(SST)受体拮抗剂，在直肠癌(CRC)细胞中通过抑制1型生长抑素受体(SSTR1)的信号传导，有效降低结细胞增殖、ALDH+细胞群体的大小以及球形成。
TP2469	Preprosomatostatin (25-34)
	Preprosomatostatin (25-34) is a peptide.
TP1570	Cortistatin-14
	Cortistatin 14 is a neuropeptide expressed in inhibitory neurons of the cerebral cortex. Depresses neuronal activity, and induces slow-wave sleep, likely through antagonism of acetylcholine. It is structurally and functionally similar to somatostatin 14.
TP2052L	CTOP acetate	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	CTOP acetate 是一种生长抑素类似物和μ-阿片受体拮抗剂。
T28743	Seglitide acetate MK 678,MK678,MK-678	Somatostatin	GPCR/G Protein
	Seglitide acetate (MK-678) 是一种选择性的 sst2生长抑素受体激动剂。
TP1570L	Cortistatin-14 acetate Cortistatin-14 acetate(186901-48-4 Free base)	Somatostatin	GPCR/G Protein
	Cortistatin-14 acetate 是一种与生长抑素-14结构相似的神经肽，通过生长抑素受体 (sst1-sst5) 结合并发挥作用。Cortistatin-14 acetate 具有抗惊厥、神经保护作用和显著的抗炎作用。
T39262L	BIM-23190 aceate	Somatostatin	GPCR/G Protein
	BIM-23190 aceate 是一种生长抑素类似物，一种 SSTR2 和 SSTR5 的选择性激动剂。 BIM-23190 可用于癌症和肢端肥大症研究。
TP1188L	Cortistatin 14, human, rat acetate	Somatostatin	GPCR/G Protein
	Cortistatin 14, human, rat acetate 是一种与 somatostatin-14 结构相似的神经肽，具有抗惊厥、神经保护作用和显着的抗炎特性。 Cortistatin 14, human, rat acetate 通过与生长抑素受体结合并发挥其功能。
T8359	Lanreotide acetate Lanreotide acetate (108736-35-2 free base),BIM 23014 (acetate),BIM 23014 acetate	Others	Others
	Lanreotide acetate (BIM 23014 acetate) 是生长抑素类似物，具有抗肿瘤活性，可用于类癌综合症。
TP1346	CYN 154806 TFA CYN 154806 TFA	Somatostatin	GPCR/G Protein
	CYN 154806 TFA(183658-72-2 free base) 是一种环状八肽，是一种有效的选择性生长抑素 sst2 受体拮抗剂。对于重组 sst2、sst1、sst3、sst4 和 sst5 受体，pIC50 值分别为 8.58、5.41、6.07、5.76 和 6.48。
T27787L	L-797,591 hydrochloride L-797,591 hydrochloride(217480-24-5 Free base)
	L-797,591 hydrochloride 对生长抑素受体亚型 1 (SSTR1)有活性。L-797,591 hydrochloride 常与 AG1478 联合使用来增强表达 SSTR1的细胞中 p-ERK5的表达。L-797,591 hydrochloride 在共转染的细胞中显著增强了 p38的磷酸化，这一作用在与 AG1478联合处理时被逆转。
TP2050L	CTAP(TFA） (103429-32-9 free base) CTAP(TFA）	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	CTAP(TFA) (103429-32-9 free base) 是一种有效的、高度选择性的、脑渗透性 μ-阿片受体拮抗剂，IC50 为 3.5 nM。它的选择性比 δ 阿片类药物 (IC50=4500 nM) 和生长抑素受体高 1200 倍以上。 CTAP TFA 可用于研究 L-DOPA 诱导的运动障碍 (LID)
T23073	NNC 26-9100	Others	Others
	Somatostatin sst4 receptor agonist
T23479	TT 232	Others	Others
	sst1/sst4 somatostatin receptors agonist
T30175	Ass 51 Ass-51,Ass51
	Ass 51 is a somatostatin analog.
T35142	Wy 40770 Wy40770,Wy-40770
	Wy 40770 is an analog of somatostatin.
T24860	TC-G1003 TC G1003
	TC-G1003 is an effective agonist of the somatostatin sst2 receptor.
T28220	NVP ACQ090 NVP-ACQ090,ACQ090,ACQ 090,NVPACQ090,ACQ-090
	NVP ACQ090 is a potent and subtype-selective somatostatin sst(3) receptor antagonist.
T40886	Onzigolide BIM-23A760,TBR-760,Onzigolide
	Onzigolide (BIM-23A760), a chimeric compound combining properties of both dopamine and somatostatin, exhibits strong agonistic activity towards the D2 subtype of dopamine receptors (D2R) as well as type 2 somatostatin receptors (SSTR2).
T69836	Paltusotine HCl
	Paltusotine, also known as CRN00808, is a somatostatin receptor agonist.

化合物

Cat.No: TP1302

Cyclic somatostatin Acetate(38916-34-6(free base))

Cat.No: TP1035L

Synonym: Somatostatin (sheep), monoacetate (salt),Somatostatin-14,SRIF-14,monoacetate (salt)

Target: Others

Somatostatin 1-28 acetate

Cat.No: TP2124L

Synonym: Somatostatin 1-28 acetate(74315-46-1 Free base)

Target: Somatostatin

Cyclic somatostatin

Cat.No: TP1035

Synonym: SRIF-14,合成生长抑素,环状生长激素抑制素,Somatostatin-14

Target: Others

Tyr-Somatostatin-14 acetate(58100-03-1 free base)

Cat.No: TP1790L

Target: Others

[Tyr11]-Somatostatin

Cat.No: T40680

Synonym: [Tyr11]-Somatostatin

[Tyr1]-Somatostatin-14

Cat.No: T40679

Synonym: [Tyr1]-Somatostatin-14

Somatostatin RC 102

Cat.No: T26200

Synonym: Somatostatin RC102,Somatostatin-RC-102,Somatostatin RC-102

Somatostatin-28 (1-12)

Cat.No: TP1258

Synonym: 1-12-Somatostatin-28,Somatostatin-28 1-12

Somatostatin-28 (1-14)

Cat.No: TP1823

Synonym: Somatostatin-28 1-14

Somatostatin-25

Cat.No: TP1810

Somatostatin 1-28

Cat.No: TP2124

Tyr-Somatostatin-14

Cat.No: TP1790

Somatostatin(3-6)

Cat.No: T34683

Synonym: Cys-lys-asn-phe

Tyr-Somatostatin-28

Cat.No: T76460

Cat.No: T2584

Synonym: SMS 201-995,奥曲肽

Target: Somatostatin

[D-Trp8,Tyr11] Somatostatin

Cat.No: T83494

Pasireotide Acetate

Cat.No: TP2207

Target: Somatostatin

[D-Trp8] Somatostatin-14

Cat.No: T83493

Cat.No: T9692

Target: Somatostatin

Cat.No: T7829

Target: Somatostatin

[Nle8] Somatostatin (1-28)

Cat.No: T76461

(D-Trp8,D-Cys14)-Somatostatin-14

Cat.No: T83546

[Tyr12] Somatostatin 28 (1-14)

Cat.No: T76459

Octreotide Acetate

Cat.No: T4119

Synonym: 醋酸奥曲肽,SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)

Target: Somatostatin

Cat.No: T20204

Synonym: 依多曲肽,SMT 487,SMT487,SMT-487

Target: Others

(D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide

Cat.No: T76612

Tyr-(D-Dab4,Arg5,D-Trp8)-cyclo-Somatostatin-14 (4-11)

Cat.No: T80135

Cat.No: TP2045

Cyclosomatostatin Acetate

Cat.No: T21567L

Synonym: Cyclosomatostatin Acetate （84211-54-1 Free base）

Target: Somatostatin

Cyclosomatostatin TFA

Cat.No: T75842

Preprosomatostatin (25-34)

Cat.No: TP2469

Cat.No: TP1570

Cat.No: TP2052L

Target: Opioid Receptor

Seglitide acetate

Cat.No: T28743

Synonym: MK 678,MK678,MK-678

Target: Somatostatin

Cortistatin-14 acetate

Cat.No: TP1570L

Synonym: Cortistatin-14 acetate(186901-48-4 Free base)

Target: Somatostatin

BIM-23190 aceate

Cat.No: T39262L

Target: Somatostatin

Cortistatin 14, human, rat acetate

Cat.No: TP1188L

Target: Somatostatin

Lanreotide acetate

Cat.No: T8359

Synonym: Lanreotide acetate (108736-35-2 free base),BIM 23014 (acetate),BIM 23014 acetate

Target: Others

Cat.No: TP1346

Synonym: CYN 154806 TFA

Target: Somatostatin

L-797,591 hydrochloride

Cat.No: T27787L

Synonym: L-797,591 hydrochloride(217480-24-5 Free base)

CTAP(TFA） (103429-32-9 free base)

Cat.No: TP2050L

Synonym: CTAP(TFA）

Target: Opioid Receptor

Cat.No: T23073

Target: Others

Cat.No: T23479

Target: Others

Cat.No: T30175

Synonym: Ass-51,Ass51

Cat.No: T35142

Synonym: Wy40770,Wy-40770

Cat.No: T24860

Synonym: TC G1003

Cat.No: T28220

Synonym: NVP-ACQ090,ACQ090,ACQ 090,NVPACQ090,ACQ-090

Cat.No: T40886

Synonym: BIM-23A760,TBR-760,Onzigolide

Paltusotine HCl

Cat.No: T69836

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