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6

抑制剂 & 化合物

6

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1158 Copper tripeptide

[N2-(N-甘氨酰-L-组氨酰)-L-赖氨酸]铜,GHK-Cu

Others; Endogenous Metabolite Metabolism; Others
Copper tripeptide (GHK-Cu) 是天然存在的三肽,首先从人血浆中分离,但也能够在唾液和尿液中发现。它能够提高成纤维细胞中胶原蛋白,弹性蛋白,蛋白多糖和糖胺聚糖中信使 RNA 的产生。在伤口愈合期间,它能够通过蛋白水解从现有的细胞外蛋白质中除去,并且用作炎性和内皮细胞的化学引诱物。它是皮肤再生中多种细胞途径的天然调节剂。
T0594 Diphenmanil methylsulfate

Diphemanil mesylate,Diphemanil Methylsulfate,甲硫二苯马尼

AChR Neuroscience
Diphenmanil methylsulfate (Diphemanil mesylate) 是一种抗胆碱能季铵盐,可与毒蕈碱乙酰胆碱受体结合,从而减少胃酸、汗液和唾液的分泌。
T73785 D-Fructose-6-phosphate

D-Fructose 6-phosphate 是存在于唾液中的内源代谢物,可用于研究路易体痴呆。
T73769 Isocitric acid

Isocitric acid,一种存在于唾液和细胞细胞质中的内源代谢物,其研究应用范围包括阿尔茨海默氏症、路易体痴呆和缺氧。
T69232 Atropine Oxide Hydrochloride

Atropine Oxide is a derivative of Atropine. Atropine is a medication to treat certain types of nerve agent and pesticide poisonings as well as some types of slow heart rate and to decrease saliva production during surgery. Atropine is a competitive antagonist of the muscarinic acetylcholine receptor types M1, M2, M3, M4 and M5. It is classified as an anticholinergic drug (parasympatholytic).
T65252 Pepsin

Pepsin is an endopeptidase that breaks down proteins into smaller peptides and amino acids that can be easily absorbed in the small intestine[1]. Pepsin is stable at pH ranges as high as pH 6. Above this pH, pepsin is rapidly irreversibly inactivated and elevation of pH of the reaction mixture to pH 8 results in complete inactivation of pepsin[2]. Pepsin has been posited to be a reliable biological marker of EER. An immunologic pepsin assay of combined sputum and saliva was determined to be 100%...

化合物

Copper tripeptide
Cat.No: TP1158
Synonym: [N2-(N-甘氨酰-L-组氨酰)-L-赖氨酸]铜,GHK-Cu
Target: Others, Endogenous Metabolite
Diphenmanil methylsulfate
Cat.No: T0594
Synonym: Diphemanil mesylate,Diphemanil Methylsulfate,甲硫二苯马尼
Target: AChR
D-Fructose-6-phosphate
Cat.No: T73785
Synonym:
Target:
Isocitric acid
Cat.No: T73769
Synonym:
Target:
Atropine Oxide Hydrochloride
Cat.No: T69232
Synonym:
Target:
Pepsin
Cat.No: T65252
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4784 (S)-(-)-Phenylethanol

(S)-(-)-1-Phenylethanol,右旋1-苯乙醇,(-)-Methyl phenyl carbinol,(S)-(-)-sec-Phenylethyl alcohol

Others; Endogenous Metabolite Metabolism; Others
(S)-(-)-Phenylethanol ((-)-Methyl phenyl carbinol) 是内源性代谢产物的一种。
Fr14438 p-Toluic Acid

对甲基苯甲酸,4-Methylbenzoic acid

Endogenous Metabolite Metabolism
p-Toluic Acid (4-Methylbenzoic acid) 是一种合成对氨基甲基苯甲酸 (PAMBA),是被取代的苯甲酸,是一种对甲苯腈等的中间体。
T4798 N-Acetyl-L-leucine

Others; Endogenous Metabolite Metabolism; Others
N-Acetyl-L-leucine 是内源性代谢产物的一种。
T4S1619 L-Hyoscyamine sulfate

Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate,硫酸天仙子胺水合物,L-莨菪碱硫酸盐

AChR Neuroscience
L-Hyoscyamine sulfate (Levsin Sulfate) 是来自山莨菪的一种托烷生物碱,是竞争性的毒蕈碱受体拮抗剂。它是 Atropine 的左旋异构体。
T5302 (R)-pyrrolidine-2-carboxylic acid

D-脯氨酸,D-Proline

Others; Endogenous Metabolite Metabolism; Others
(R)-pyrrolidine-2-carboxylic acid (D-Proline) 是天然氨基酸 L -脯氨酸的异构体。D -氨基酸在人类血浆和唾液中含量相对较高。这些氨基酸可能是细菌来源,但也有证据表明它们是通过氨基酸消旋酶活性内源性产生的。
T0962 L-Hyoscyamine

Daturine,Hyoscyamine,L-莨菪碱,L-天仙子胺

AChR Neuroscience
L-Hyoscyamine (Daturine) 是从山莨菪中提取的一种托烷生物碱,是竞争性的毒蕈碱受体拮抗剂。它是 Atropine 的左旋异构体。

天然产物

(S)-(-)-Phenylethanol
Cat.No: T4784
Synonym: (S)-(-)-1-Phenylethanol,右旋1-苯乙醇,(-)-Methyl phenyl carbinol,(S)-(-)-sec-Phenylethyl alcohol
Target: Others, Endogenous Metabolite
p-Toluic Acid
Cat.No: Fr14438
Synonym: 对甲基苯甲酸,4-Methylbenzoic acid
Target: Endogenous Metabolite
N-Acetyl-L-leucine
Cat.No: T4798
Synonym:
Target: Others, Endogenous Metabolite
L-Hyoscyamine sulfate
Cat.No: T4S1619
Synonym: Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate,硫酸天仙子胺水合物,L-莨菪碱硫酸盐
Target: AChR
(R)-pyrrolidine-2-carboxylic acid
Cat.No: T5302
Synonym: D-脯氨酸,D-Proline
Target: Others, Endogenous Metabolite
L-Hyoscyamine
Cat.No: T0962
Synonym: Daturine,Hyoscyamine,L-莨菪碱,L-天仙子胺
Target: AChR
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