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Cat. No. Product Name Target Signaling Pathways
T61972 Pomaglumetad methionil hydrochloride

LY2140023 hydrochloride

GluR Neuroscience
Pomaglumetad methionil hydrochloride (LY2140023 hydrochloride) (LY2140023 hydrochloride) 是的 LY404039 的蛋氨酸前药,具有口服活性。LY404039是一种选择性 mGlu2/3 受体激动剂。Pomaglumetad methionil hydrochloride 可用于精神分裂症的研究。
T6022 LY404039

pomaglumetad

Glucocorticoid Receptor; GluR Endocrinology/Hormones; Neuroscience
LY404039 (pomaglumetad) 是可口服的mGluR2和mGluR3选择性激动剂,有抗精神病和抗焦虑的作用。它对重组人mGluR2和mGluR3的Ki 分别为 149 和 92 nM,比对其他受体/转运蛋白的抑制性高 100 倍以上。
T12520 Pomaglumetad methionil

LY2140023 hydrate

GluR Neuroscience
Pomaglumetad methionil is an oral methionine prodrug of the potent specific agonist of mGlu2/3 receptor LY404039.
T11907 Pomaglumetad methionil anhydrous

LY2140023

GluR Neuroscience
LY2140023 has the potential for schizophrenia.LY2140023 is an orally active prodrug of LY404039. LY404039 is a selective metabotropic glutamate 2/3 receptor agonist.

化合物

Pomaglumetad methionil hydrochloride
Cat.No: T61972
Synonym: LY2140023 hydrochloride
Target: GluR
LY404039
Cat.No: T6022
Synonym: pomaglumetad
Target: Glucocorticoid Receptor, GluR
Pomaglumetad methionil
Cat.No: T12520
Synonym: LY2140023 hydrate
Target: GluR
Pomaglumetad methionil anhydrous
Cat.No: T11907
Synonym: LY2140023
Target: GluR
TargetMol Loading
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