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6

抑制剂 & 化合物

6

天然产物

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Cat. No. Product Name Target Signaling Pathways
T20958 Hexazinone

Others Others
Hexazinone 是三嗪家族的广谱除草剂。 Hexazinone 通过与光系统 II 中电子传递链的 D-1 醌蛋白结合来抑制光合作用。
T5117 Hexaflumuron

Others Others
Hexazinone 是一种三嗪家族的非选择性除草剂。它能够同光系统 II 电子传递链的 D-1 醌蛋白结合,抑制光合作用的发生。
TD0104 Methyl purple

Others Others
Methyl purple 是一种引入的醌-酰亚胺氧化还原染料,已被证明是一种对叶绿体中光系统 I 活性异常敏感的监测器。
T74695 Antimalarial agent 17

Antimalarial agent 17,一种兼具抗疟和除草功能的化合物,作为光系统 II 型抑制剂,在出苗后除草活性方面与市售除草剂表现出相当的效力。
T14218 Amicarbazone

BAY314666,胺唑草酮,BAY-MKH 3586

Others Others
Amicarbazone (BAY-MKH3586; BAY314666) is a potent PSII inhibitor, disrupting photosynthetic electron transport by binding to the Qb domain of photosystem II. This broad-spectrum herbicide is effective through foliar and root application, showcasing rapid absorption and translocation. However, its effectiveness can be compromised by common PSII inhibitor resistance. With an IC50 value indicating high potency, amicarbazone leads to chlorosis, stunted growth, tissue necrosis, and death in sensitive...
T82635 Cy-FBP/SBPase-IN-1

Cy-FBP/SBPase-IN-1(compound S5)是一种针对蓝藻光合作用调节酶的Cy-FBP/SBPase抑制剂。该化合物能有效阻断卡尔文循环和光系统,从而减少蓝藻的光合效率。此外,Cy-FBP/SBPase-IN-1能抑制包括集胞藻PCC6803在内的蓝藻生长,并在人源细胞与斑马鱼模型中表现出良好的安全性。

化合物

Hexazinone
Cat.No: T20958
Synonym:
Target: Others
Hexaflumuron
Cat.No: T5117
Synonym:
Target: Others
Methyl purple
Cat.No: TD0104
Synonym:
Target: Others
Antimalarial agent 17
Cat.No: T74695
Synonym:
Target:
Amicarbazone
Cat.No: T14218
Synonym: BAY314666,胺唑草酮,BAY-MKH 3586
Target: Others
Cy-FBP/SBPase-IN-1
Cat.No: T82635
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5080 Spermidine trihydrochloride

Spermidine hydrochloride,4-Azaoctamethylenediamine trihydrochloride,三盐酸亚精胺,亚精胺盐酸盐

NMDAR; Autophagy Autophagy; Neuroscience
Spermidine trihydrochloride (4-Azaoctamethylenediamine trihydrochloride) 能够维持细胞膜稳定性,提高抗氧化酶特性,改善光系统 II (PSII) 以及相关基因表达,也能够显著抑制 H2O2和 O2.-含量。
T4893 Spermidine

N-(3-Aminopropyl)-1,4-diaminobutane,亚精胺,N-(4-Aminobutyl)-1,3-diaminopropane

Endogenous Metabolite Metabolism
Spermidine (N-(3-Aminopropyl)-1,4-diaminobutane) 能够维持细胞膜稳定性,提高抗氧化酶活性,改善光系统 II 以及相关基因表达。它结合并激活 NMDA,并已显示以浓度依赖性方式增强 NMDA 诱导的电流。
T81158 Siderin

Siderin作为一种Photosystem II抑制剂,有效地阻断了离体菠菜光合过程中ATP的合成及叶绿体电子传递,因此被用于植物光合作用的研究。
TN3557 Cabraleadiol

ATPase; Antifection Membrane transporter/Ion channel; Microbiology/Virology
Cabraleadiol displays antimycobacterial activity against Mycobacterium tuberculosis, it also is weakly cytotoxic to a breast cancer (BC) cell line. Cabraleadiol inhibits photosystem II (PS II) and induces the appearance of small G band which is related wi
T17037 Tenuazonic acid

Others Others
Tenuazonic acid is a putative nonhost-selective mycotoxin isolated from Alternaria alternate. Tenuazonic acid blocks electron transport beyond primary quinone acceptor (QA) by interacting with D1 protein and it is a broad-spectrum and effective photosyste
TN3930 Encecalin

ATPase Membrane transporter/Ion channel
Encecalin and demethylencecalin are major phytotoxic compounds isolated from Helianthella quinquenervis (Hook) A Gray (Asteraceae), they inhibit photosystem II (from water to 2,5-dibromo-3-methyl-6-isopropyl-1,4 p-benzo-quinone).They retard seed germinati

天然产物

Spermidine trihydrochloride
Cat.No: T5080
Synonym: Spermidine hydrochloride,4-Azaoctamethylenediamine trihydrochloride,三盐酸亚精胺,亚精胺盐酸盐
Target: NMDAR, Autophagy
Spermidine
Cat.No: T4893
Synonym: N-(3-Aminopropyl)-1,4-diaminobutane,亚精胺,N-(4-Aminobutyl)-1,3-diaminopropane
Target: Endogenous Metabolite
Siderin
Cat.No: T81158
Synonym:
Target:
Cabraleadiol
Cat.No: TN3557
Synonym:
Target: ATPase, Antifection
Tenuazonic acid
Cat.No: T17037
Synonym:
Target: Others
Encecalin
Cat.No: TN3930
Synonym:
Target: ATPase
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