Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15275 |
Fenobam
|
GluR | Neuroscience |
Fenobam 是可口服的、可穿过血脑屏障的 mGluR5拮抗剂,具有抗焦虑活性,在大鼠和人重组 mGlu5 受体上的 Kd 值分别 54 和 31 nM。它有反向激动剂活性,可阻断 mGlu5 受体活性,IC50为 84 nM。 | |||
T4688 |
Pipequaline hydrochloride
PK-8165 hydrochloride,盐酸哌夸林 |
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
Pipequaline hydrochloride (PK-8165 hydrochloride) 是一种苯二氮卓受体部分激动剂,有抗焦虑作用。 | |||
T12763 | Ro 41-3290 | Others | Others |
Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor. | |||
T24367 |
Y 23684
Y23684,Y-23684 |
||
Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic. | |||
T4655 |
Pipequaline
PK-8165,哌夸林 |
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
Pipequaline (PK-8165) 是一种苯二氮卓受体部分激动剂,有抗焦虑作用。 |