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Cat. No. Product Name Target Signaling Pathways
T79321 nSMase2-IN-1

Phospholipase Metabolism
nSMase2-IN-1是一款口服活性的nSMase2抑制剂,具有0.13 ± 0.06 μM的IC50。该化合物在肝脏微粒体内具有良好的代谢稳定性,口服给药后获得较高的脑血浆比值,适用于神经系统疾病研究。
T4985 Neticonazole Hydrochloride

Antifungal Microbiology/Virology
Neticonazole hydrochloride 是一种咪唑衍生物,具有抗感染和抗癌作用。它也是一种长效抗真菌剂。
T69756 GT-2331

GT-2331 is a histamine H3 receptor antagonist.
T69757 PDDC inhibitor

PDDC is the first nSMase2 inhibitor that possesses both favorable pharmacodynamics and pharmacokinetic (PK) parameters, including substantial oral bioavailability, brain penetration, and significant inhibition of exosome release from the brain in vivo.

化合物

nSMase2-IN-1
Cat.No: T79321
Synonym:
Target: Phospholipase
Neticonazole Hydrochloride
Cat.No: T4985
Synonym:
Target: Antifungal
GT-2331
Cat.No: T69756
Synonym:
Target:
PDDC inhibitor
Cat.No: T69757
Synonym:
Target:
TargetMol Loading
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