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Cat. No. Product Name Target Signaling Pathways
T22062 CCG-100602

Rho; Ras Cell Cycle/Checkpoint; GPCR/G Protein; MAPK
CCG-100602 是心肌蛋白相关转录因子 A/血清反应因子信号转导的特异性抑制剂。它抑制 PC-3 前列腺癌细胞中 RhoA/C 介导的、SRF 驱动的荧光素酶表达,IC50为 9.8 µM。
T7764 CCG-222740

ROCK; Rho; Ras Cell Cycle/Checkpoint; Cytoskeletal Signaling; GPCR/G Protein; MAPK; Stem Cells
CCG-222740 是一种口服有效的选择性Rho/MRTF 途径抑制剂。它也是 α-平滑肌的肌动蛋白表达抑制剂,可减少皮肤纤维化并阻止黑色素瘤转移。
T68431 CCG-58150

CCG-58150 is a potentiInhibitor of Rho/Myocardin-Related Transcription Factor (MRTF)/Serum Response Factor (SRF)-Mediated Gene Transcription as Potential Antifibrotic Agents for Scleroderma.
T23296 (S)-CCG-1423

Others Others
(S)-CCG-1423 is a stereoisomer of CCG-1423. CCG-1423 is a Rho inhibitor involved in blocking signaling through myocardin-related transcription factor A and serum response factor.
T23221 (R)-CCG-1423

Others Others
(R)-CCG-1423 is a stereoisomer of CCG-1423. CCG-1423 is a Rho inhibitor involved in blocking signaling through myocardin-related transcription factor A (MRTF-A) and serum response factor (SRF).

化合物

CCG-100602
Cat.No: T22062
Synonym:
Target: Rho, Ras
CCG-222740
Cat.No: T7764
Synonym:
Target: ROCK, Rho, Ras
CCG-58150
Cat.No: T68431
Synonym:
Target:
(S)-CCG-1423
Cat.No: T23296
Synonym:
Target: Others
(R)-CCG-1423
Cat.No: T23221
Synonym:
Target: Others
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