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5

抑制剂 & 化合物

5

天然产物

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Cat. No. Product Name Target Signaling Pathways
T3158L Harman hydrochloride

哈尔满盐酸盐,Harmane hydrochloride(486-84-0 Free base)

P450 Metabolism
Harman hydrochloride 可以以 AhR 依赖性方式直接诱导 CYP1A1 基因表达,可能代表了harman 促进致突变性、共致突变性和致癌性的新机制。
T5941 Anthraflavic acid

2,6-二羟基蒽醌,2,6-Dihydroxyanthraquinone

Others Others
Anthraflavic acid (2,6-Dihydroxyanthraquinone) 是一种特异性细胞色素 P-448抑制剂,细胞色素 P-448 是与许多化学致癌物质的激活密切相关的酶系统。它是一种类黄酮,有效的IQ 诱变性抑制剂,能够抑制微粒体和胞质激活途径。
T0770 Carbadox

Getroxel,卡巴多,Mecadox

Antibacterial; Antibiotic Microbiology/Virology
Carbadox (Mecadox) 是一种喹喔啉二氧化氮抗生素,用于育龄期的猪,治疗猪痢疾和肠炎,促进成长。
TD0002L CelRed nucleic acid gel stain *10,000× concentrate in DMSO*

1) Non-toxicity: The unique oiliness and high molecular weight characteristics of CelRed prevent it from penetrating cell membranes into cells. Ames test results also show that the mutagenicity of CelRed dye is much less than that of EB. 2) High sensitivi
TD0002 CelRed nucleic acid gel stain *10,000× concentrate in water*

1) Non-toxicity: The unique oiliness and high molecular weight characteristics of CelRed prevent it from penetrating cell membranes into cells, and Ames test results also show that the mutagenicity of CelRed dye is much less than EB. 2) High sensitivity:

化合物

Harman hydrochloride
Cat.No: T3158L
Synonym: 哈尔满盐酸盐,Harmane hydrochloride(486-84-0 Free base)
Target: P450
Anthraflavic acid
Cat.No: T5941
Synonym: 2,6-二羟基蒽醌,2,6-Dihydroxyanthraquinone
Target: Others
Carbadox
Cat.No: T0770
Synonym: Getroxel,卡巴多,Mecadox
Target: Antibacterial, Antibiotic
CelRed nucleic acid gel stain *10,000× concentrate in DMSO*
Cat.No: TD0002L
Synonym:
Target:
CelRed nucleic acid gel stain *10,000× concentrate in water*
Cat.No: TD0002
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T19081 1,3-Dithiane

1,3-Dithian,M-DITHIANE,1,3-Dithiacyclohexane,1,3-二噻烷

Anti-infection; Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
1,3-Dithiane (1,3-Dithian) 是一种受保护的甲醛阴离子等价物,可用作有用的标记合成子。它是在煮熟的牛肉提取物中发现的含硫美拉德反应产物 。
TL0013 Heraclenin

独活内酯

Anti-infection; Immunology/Inflammation related Immunology/Inflammation; Microbiology/Virology
Heraclenin 是一种天然呋喃香豆素。它浓度依赖性的靶向激活的 T 细胞核因子 (NFAT) ,抑制人原代 T 细胞中 T 细胞受体介导的增殖。
TN1084 1,3,5,8-Tetrahydroxyxanthone

Desmethylbellidifolin,去甲基雏叶龙胆酮

Anti-infection Microbiology/Virology
1,3,5,8-Tetrahydroxyxanthone (Desmethylbellidifolin) 是一种天然黄酮,从 Gentianella acuta 中提取得到。它具有镇痉作用和抗炎作用。
T4715 2'-Deoxyguanosine monohydrate

2'-脱氧鸟苷一水合物,Guanine-2'-deoxyriboside

Others; Endogenous Metabolite Metabolism; Others
2'-Deoxyguanosine monohydrate (Guanine-2'-deoxyriboside) 是内源性代谢产物的一种。
TN4928 Rutacridone

P450 Metabolism
Rutacridone has mutagenicity.

天然产物

1,3-Dithiane
Cat.No: T19081
Synonym: 1,3-Dithian,M-DITHIANE,1,3-Dithiacyclohexane,1,3-二噻烷
Target: Anti-infection, Endogenous Metabolite, Antibacterial
Heraclenin
Cat.No: TL0013
Synonym: 独活内酯
Target: Anti-infection, Immunology/Inflammation related
1,3,5,8-Tetrahydroxyxanthone
Cat.No: TN1084
Synonym: Desmethylbellidifolin,去甲基雏叶龙胆酮
Target: Anti-infection
2'-Deoxyguanosine monohydrate
Cat.No: T4715
Synonym: 2'-脱氧鸟苷一水合物,Guanine-2'-deoxyriboside
Target: Others, Endogenous Metabolite
Rutacridone
Cat.No: TN4928
Synonym:
Target: P450
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