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Cat. No. Product Name Target Signaling Pathways
T10831L Cl-amidine hydrochloride

Apoptosis; PAD Apoptosis; Chromatin/Epigenetic
Cl-amidine hydrochloride 是一种口服有效的PAD 抑制剂,可阻断组蛋白 3 瓜氨酸化和中性粒细胞胞外陷阱的形成,并提高败血症小鼠的存活率。它可诱导癌细胞凋亡,还可诱导 miR-16 引起细胞周期阻滞。
T10831 Cl-amidine

Others Others
Cl-amidine is an orally active inhibitor of peptidyl arginine deminase (PAD) (IC50s: 0.8 μM, 6.2 μM, and 5.9 μM for PAD1, PAD3, and PAD4). Cl-amidine induces apoptosis in cancer cells.
T10831L2 Cl-amidine TFA

Others Others
Cl-amidine TFA is an orally active inhibitor of peptidyl arginine deminase (PAD) (IC50s: 0.8 μM, 6.2 μM, and 5.9 μM for PAD1, PAD3, and PAD4). Cl-amidine induces apoptosis in cancer cells.

化合物

Cl-amidine hydrochloride
Cat.No: T10831L
Synonym:
Target: Apoptosis, PAD
Cl-amidine
Cat.No: T10831
Synonym:
Target: Others
Cl-amidine TFA
Cat.No: T10831L2
Synonym:
Target: Others
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