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Cat. No. Product Name Target Signaling Pathways
T14141 AGI-24512

Others; Methionine Adenosyltransferase (MAT) Chromatin/Epigenetic; Others
AGI-24512 是一种甲硫氨酸腺苷转移酶 2A 抑制剂,在体外能够阻断 MTAP 缺失的癌细胞的生长,可用于研究癌症。
TQ0008 MT-DADMe-ImmA

Methylthio-DADMe-Immucillin A,MTDIA

Others Others
MT-DADMe-ImmA (MTDIA) 是一种人5'-甲硫基腺苷磷酸化酶的抑制剂 (MTAP)(Ki:90 pM)。
T12908 SIBA

5'-Deoxy-5'-isobutylthioadenosine,5'-Isobutylthioadenosine,5ˊ-异丁硫基-5ˊ-脱氧腺苷

Nucleoside Antimetabolite/Analog; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
SIBA (5'-Deoxy-5'-isobutylthioadenosine) 是 SAH 的合成类似物,可作为 S-腺苷甲硫氨酸介导的甲基转移的抑制剂。它干扰多种酶活性,可逆地阻断单纯疱疹病毒 1 型病毒的繁殖。
T31672 Erythrofuranosyladenine

9-β-D-Erythrofuranosyladenine,ETA

Erythrofuranosyladenine(9-beta-D-Erythrofuranosyladenine, ETA) is a nontoxic MTAP substrate. Erythrofuranosyladenine is an effective salvage agent for methylthioadenosine phosphorylase–selective therapy of T-cell acute lymphoblastic leukemia with L-alanos

化合物

AGI-24512
Cat.No: T14141
Synonym:
Target: Others, Methionine Adenosyltransferase (MAT)
MT-DADMe-ImmA
Cat.No: TQ0008
Synonym: Methylthio-DADMe-Immucillin A,MTDIA
Target: Others
SIBA
Cat.No: T12908
Synonym: 5'-Deoxy-5'-isobutylthioadenosine,5'-Isobutylthioadenosine,5ˊ-异丁硫基-5ˊ-脱氧腺苷
Target: Nucleoside Antimetabolite/Analog, HSV
Erythrofuranosyladenine
Cat.No: T31672
Synonym: 9-β-D-Erythrofuranosyladenine,ETA
Target:
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