Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10777 |
CG347B
|
HDAC | Chromatin/Epigenetic; DNA Damage/DNA Repair |
CG347B 是一种选择性HDAC6抑制剂。 | |||
T0515 |
Tioxolone
|
Carbonic Anhydrase | Metabolism |
Tioxolone 是一种金属酶碳酸酐酶 I 抑制剂,具有抗痤疮作用。 | |||
T60278 |
Tyrosinase-IN-2
|
Tyrosinase | Proteases/Proteasome |
Tyrosinase-IN-2 (compound 67) 是一种有效的酪氨酸酶抑制剂。酪氨酸酶是一种含铜金属酶,负责黑色素生物合成和酶促褐变中的限速催化步骤。Tyrosinase-IN-2 具有研究皮肤美白剂和食品防腐剂的潜力。 | |||
T26298 |
ts-SA
tsSA |
||
ts-SA is a metalloenzyme carbonic anhydrase (CA) inhibitor. It is active against 7 out of 10 human CA isoforms. | |||
T61460 | Tyrosinase-IN-3 | ||
Tyrosinase-IN-3 (compound 54) is a powerful tyrosinase inhibitor, an enzyme involved in the key catalytic step of melanin biosynthesis and enzymatic browning. As a copper-containing metalloenzyme, tyrosinase plays a crucial role in these processes. The compound shows promise for studying skin whitening agents and food preservatives [1]. | |||
T76013 | Carbonic anhydrase | ||
Carbonic anhydrase 是原核生物和真核生物中普遍存在的含锌金属酶。Carbonic anhydrase 可以催化二氧化碳可逆地转化为碳酸氢盐和质子。Carbonic anhydrase 可用于癌症、青光眼、肥胖症和癫痫症的研究。 | |||
T76150 | Galactose oxidase | ||
Galactose oxidase (GOase) 半乳糖氧化酶来自真菌,常用于生化研究。Galactose oxidase 是一种 II 型铜金属酶,含有单一多肽。Galactose oxidase 催化伯醇的双电子氧化生成相应的醛,并将二氧还原为过氧化氢。 |