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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T38192 Unifiram

Others Others
Unifiram 是一种认知增强剂。 Unifiram 诱导大鼠海马 CA1 区场兴奋性突触后电位 (fEPSP) 幅度的持久增加 (EC50= 27 nM) 并增加大鼠大脑皮层中乙酰胆碱 (ACh) 的释放。
T71142 Tebuconazole-d9

Tebuconazole-d9 is intended for use as an internal standard for the quantification of tebuconazole by GC- or LC-MS. Tebuconazole is a triazole fungicide that is active against both seed and foliar fungi. It inhibits 14α-demethylase isolated from U. maydis and S. bicolor with IC50 values of 0.05 and 0.16 nM, respectively. It inhibits the androgenic effect of the androgen receptor agonist DHT (IC20 = 2.89 µM) and is cytotoxic (EC20 = 38.9 µM) in an MDA-kb2 assay. Tebuconazole (50 and 100 mg/kg per...

化合物

Unifiram
Cat.No: T38192
Synonym:
Target: Others
Tebuconazole-d9
Cat.No: T71142
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2230 Paeoniflorin

芍药苷,Peoniflorin

HSP; COX Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; Neuroscience
Paeoniflorin (Peoniflorin) 是从芍药根中提取的一种蒎烷单萜糖苷,具有抗癌作用、抗氧化应激、抗血小板聚集、血管扩张、降低血液粘度和抗炎活性等多种生物活性。它是一种热休克蛋白诱导剂,通过自噬途径保护 PC12 细胞免受 MPP+和酸性损伤。

天然产物

Paeoniflorin
Cat.No: T2230
Synonym: 芍药苷,Peoniflorin
Target: HSP, COX
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