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抑制剂 & 化合物

23

天然产物

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Cat. No. Product Name Target Signaling Pathways
T83764 Sulfane Sulfur Probe 4

​SSP4

Sulfane sulfur probe 4 (SSP4) 是用于检测含硫化氢衍生的多硫化物、过硫化物和硫化物的荧光探针。在含硫磺物种存在下,SSP4 经核苷酸攻击反应生成荧光素,其激发/发射峰值分别为494/515 nm,以及两分子的1,2-苯并二硫杂环-3-酮。SSP4 已应用于确定H2S3在原代小鼠神经元中的定位,并检测L. japonicus 幼苗根部的多硫化物。

化合物

Sulfane Sulfur Probe 4
Cat.No: T83764
Synonym: ​SSP4
Target:
Cat. No. Product Name Target Signaling Pathways
TN4661 Nodosin

IL Receptor; Autophagy Autophagy; Immunology/Inflammation
Nodosin 是一种二萜化合物,从Isodon trichocarpusKudo 和I. JaponicusHARA 中提取得到。
T3S1250 Ophiogenin 3-O-α-L-rhamnopyranosyl-(1→2)-β-D-glucopyranoside

麦冬苷元-3-O-Α-L-吡喃鼠李糖基(1→2)-Β-D-吡喃葡萄糖苷,Ophiogenin-3-O-alpha-L-rhaMnopyranosyl-(1->2)-beta-D-glucopyranoside

Others Others
Ophiogenin 3-O-α-L-rhamnopyranosyl-(1→2)-β-D-glucopyranoside (Ophiogenin-3-O-alpha-L-rhaMnopyranosyl-(1->2)-beta-D-glucopyranoside) 是一种从麦冬根中取得的萜类糖苷,对心血管系统有良好的药理作用。
TN7228 11-oxo-alpha-amyrin

Neoilexonol

11-oxo-alpha-amyrin (Neoilexonol) 是一种从Leonurus japonicus (Lamiaceae) 提取出的三萜化合物,是一种天然化合物 。
TN7110 Ginsenoside Rs2

人参皂苷Rs2

Others Others
Ginsenoside Rs2 是从人参Panax japonicus var.叶中分离得到的天然产物。
T4244 Methylophiopogonone A

Others Others
Methylophiopogonone A 是一种异黄酮,从 Ophiopogon japonicas 根部分离得到,具有抗炎作用。
T4S1247 14-Hydroxy sprengerinin C

14-羟基麦冬皂苷C,14-羟基麦冬皂苷 C

Others Others
14-Hydroxy sprengerinin C 是一种甾体化合物,提取自麦冬。
TWS1977 Kamebakaurin

尾叶香茶菜丙素,Kamebakaurine

NF-κB NF-κB
Kamebakaurin (Kamebakaurine) 是一种提取自Isodon japonicus 中的天然产物,是一种NF-κB 的抑制剂,能够抑制 p50 的 DNA 结合活性。
T81408 Preleoheterin

Preleoheterin(化合物3)为一类从L. japonicus分离得到的拉丹烷二萜。
T33641 Neoxaline

Nedoxaline

Neoxaline is an alkaloid isolated from fermentation broth of Aspergillus japonicus.
TN5010 Shizukaol A

Others Others
Shizukaol A is a natural product from Chloranthus japonicus.
T3S1253 Cixiophiopogon A

Others Others
Cixiophiopogon A is a natural product from Ophiopogon japonicus.
T83568 (25R)-Ruscogenin-3-yl α-L-rhamnopyranosyl-(1→2)-[β-D-xylopyranosyl-(1→4)]-β-D-glucopyranoside

(25R)-Ruscogenin-3-yl α-L-rhamnopyranosyl-(1→2)-[β-D-xylopyranosyl-(1→4)]-β-D-glucopyranoside (compound 1) 为源自麦冬须 (Ophiopogon japonicus) 根的甾体皂苷。
T83266 6-Formyl-isoophiopogonanone B

6-Formyl-isoophiopogonanone B,一种同型异黄酮,源自麦冬(Ophiopogon japonicus)。
T81166 Shizukaol G

Shizukaol G为一种从Chloranthus japonicus根部分离得到的二聚倍半萜烯。
T83271 6-Aldehydoisoophiopogonone B

6-Aldehydoisoophiopogonone B (Compound 24) 是从Ophiopogon japonicus 提取的同型异黄酮化合物。
TN4306 Isoleojaponin

Others Others
Isoleojaponin is a natural product from Leonurus japonicus.
TN1304 6-Formyl-isoophiopogonanone A

6-甲酰基-异沿阶草酮 A,6-Aldehydoisoophiopogonanone A,6-醛基异麦冬黄烷酮A

Others Others
6-Aldehydoisoophiopogonanone A is a natural product from Ophiopogon japonicus.
T81167 Shizukanolide

Shizukanolide,一种倍半萜内酯,源自金兰属 (Chloranthus japonicus) 植物,其脱氢衍生物展现出中等抗真菌活性。
TN6231 3,4-Dihydroxyallylbenzene 3,4-di-O-glucoside

1,2-Di-O-β-D-glucopyranosyl-4-allylbenzene

Others Others
3,4-Dihydroxyallylbenzene 3,4-di-O-glucoside (1,2-Di-O-β-D-glucopyranosyl-4-allylbenzene) 是一种在麦冬块茎中发现的天然产物。
T82487 Ejaponine A

Ejaponine A(化合物1)为源于日本卫矛的杀虫倍半萜酯。该化合物展现出强效针对粘虫的活性(LD50为89.2 μg/g),在相关杀粘虫机制研究中得到应用。
T13805 Ophiopogonin C

Ophiopogonin C,麦冬胶原蛋白 C

Others Others
Ophiopogonin C is a natural product isolated from the tubers of Ophiopogon japonicus, is a rare naturally occurring C29 steroidal glycoside.
T81601 Ophiopogonone C

Ophiopogonone C(化合物3),一异黄酮类化合物,自麦冬块茎乙醇提取物中分离。
T37609 (rel)-Asperparaline A

Aspergillimide is a fungal metabolite originally isolated from A. japonicus.1 It reduces nicotinic acetylcholine receptor (nAChR) peak and slowly-desensitizing amplitudes induced by acetylcholine in silkworm (B. mori) larval neurons (IC50s = 20.2 and 39.6 nM, respectively) but has no effect on chicken α3β4-, α4β2-, and α7-containing nAChRs.2 Dietary administration of aspergillimide A (10 μg/g of diet) induces paralysis in silkworm fourth instar larvae.1 Aspergillimide A (10 and 20 mg/kg) reduces...

天然产物

Nodosin
Cat.No: TN4661
Synonym:
Target: IL Receptor, Autophagy
Ophiogenin 3-O-α-L-rhamnopyranosyl-(1→2)-β-D-glucopyranoside
Cat.No: T3S1250
Synonym: 麦冬苷元-3-O-Α-L-吡喃鼠李糖基(1→2)-Β-D-吡喃葡萄糖苷,Ophiogenin-3-O-alpha-L-rhaMnopyranosyl-(1->2)-beta-D-glucopyranoside
Target: Others
11-oxo-alpha-amyrin
Cat.No: TN7228
Synonym: Neoilexonol
Target:
Ginsenoside Rs2
Cat.No: TN7110
Synonym: 人参皂苷Rs2
Target: Others
Methylophiopogonone A
Cat.No: T4244
Synonym:
Target: Others
14-Hydroxy sprengerinin C
Cat.No: T4S1247
Synonym: 14-羟基麦冬皂苷C,14-羟基麦冬皂苷 C
Target: Others
Kamebakaurin
Cat.No: TWS1977
Synonym: 尾叶香茶菜丙素,Kamebakaurine
Target: NF-κB
Preleoheterin
Cat.No: T81408
Synonym:
Target:
Neoxaline
Cat.No: T33641
Synonym: Nedoxaline
Target:
Shizukaol A
Cat.No: TN5010
Synonym:
Target: Others
Cixiophiopogon A
Cat.No: T3S1253
Synonym:
Target: Others
(25R)-Ruscogenin-3-yl α-L-rhamnopyranosyl-(1→2)-[β-D-xylopyranosyl-(1→4)]-β-D-glucopyranoside
Cat.No: T83568
Synonym:
Target:
6-Formyl-isoophiopogonanone B
Cat.No: T83266
Synonym:
Target:
Shizukaol G
Cat.No: T81166
Synonym:
Target:
6-Aldehydoisoophiopogonone B
Cat.No: T83271
Synonym:
Target:
Isoleojaponin
Cat.No: TN4306
Synonym:
Target: Others
6-Formyl-isoophiopogonanone A
Cat.No: TN1304
Synonym: 6-甲酰基-异沿阶草酮 A,6-Aldehydoisoophiopogonanone A,6-醛基异麦冬黄烷酮A
Target: Others
Shizukanolide
Cat.No: T81167
Synonym:
Target:
3,4-Dihydroxyallylbenzene 3,4-di-O-glucoside
Cat.No: TN6231
Synonym: 1,2-Di-O-β-D-glucopyranosyl-4-allylbenzene
Target: Others
Ejaponine A
Cat.No: T82487
Synonym:
Target:
Ophiopogonin C
Cat.No: T13805
Synonym: Ophiopogonin C,麦冬胶原蛋白 C
Target: Others
Ophiopogonone C
Cat.No: T81601
Synonym:
Target:
(rel)-Asperparaline A
Cat.No: T37609
Synonym:
Target:
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