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Cat. No. Product Name Target Signaling Pathways
T36526 IL-17 modulator 4

Interleukin Immunology/Inflammation
IL-17 modulator 4 是 IL-17 modulator 1 的前药,IL-17 modulator 1 是 IL-17 的有效调节剂。
T4050 GSK2981278

ROR gama modulator 1

ROR Metabolism
GSK2981278 (ROR gama modulator 1) 是 RORγ的选择性反向激动剂。它能够抑制 il17启动子的激活,并且干扰 RORγ-DNA 结合。
T40127 IL-17 modulator 3

IL-17 modulator 3 (US20200247785A1) is a chemical compound that acts as an IL-17 modulator. It has potential applications in researching inflammation, cancer, and autoimmune diseases.
T40106 IL-17 modulator 1

IL-17 modulator 1 is an orally active small molecule. It is highly efficacious in modulating IL-17 and can effectively prevent, treat, or ameliorate various diseases such as psoriasis, ankylosing spondylitis, and psoriatic arthritis.
T36525 IL-17 modulator 1 disodium

IL-17 Modulator 1 (disodium) is a potent, orally active compound, known for its high efficacy in modulating IL-17. This compound is extensively utilized for researching various diseases such as psoriasis, ankylosing spondylitis, and psoriatic arthritis[1].
T40107 IL-17 modulator 4 sulfate

IL-17 modulator 4 sulfate is a prodrug of IL-17 modulator 1 . IL-17 modulator 1 is an orally active, highly efficacious IL-17 modulator.
T4670 SR0987

ROR Metabolism
SR0987是SR1078 的类似物,是RORγt 的激动剂,其EC50=800 nM。它可上调IL17 的表达,并且抑制PD-1 的表达。

化合物

IL-17 modulator 4
Cat.No: T36526
Synonym:
Target: Interleukin
GSK2981278
Cat.No: T4050
Synonym: ROR gama modulator 1
Target: ROR
IL-17 modulator 3
Cat.No: T40127
Synonym:
Target:
IL-17 modulator 1
Cat.No: T40106
Synonym:
Target:
IL-17 modulator 1 disodium
Cat.No: T36525
Synonym:
Target:
IL-17 modulator 4 sulfate
Cat.No: T40107
Synonym:
Target:
SR0987
Cat.No: T4670
Synonym:
Target: ROR
TargetMol Loading
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