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55

抑制剂 & 化合物

2

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Cat. No. Product Name Target Signaling Pathways
TP2384L Hexapeptide-10 Acetate

Hexapeptide-10 Acetate(146439-94-3 Free base)

Integrin Cytoskeletal Signaling
Hexapeptide-10 Acetate (Hexapeptide-10 Acetate) 是一种合成肽。它增加层粘连蛋白 V 和 α6-整合素的合成以促进细胞结合,具有非凡的可见皮肤重组和紧致能力。
TP2492 Hexapeptide-9 Acetate

Hexapeptide-9 Acetate(1228371-11-6 Free base)

Others Others
Hexapeptide-9 Acetate 是一种胶原蛋白肽,通过与皮肤细胞自然相互作用来帮助强化结构组织,从而促进再生过程。
T8953L Acetyl hexapeptide 38 Acetate

Acetyl hexapeptide 38 Acetate(1400634-44-7 free base)

Others Others
Acetyl hexapeptide 38 Acetate(1400634-44-7 free base) 丰胸肽,是一种乙酰化六肽,能显着刺激脂肪合成部位的使用,增加胸部或脸颊的体积,塑造完美身材。
TP2490 Palmitoyl Hexapeptide-12 Acetate

Palmitoyl Hexapeptide-12 Acetate(171263-26-6 Free base)

Others Others
Palmitoyl Hexapeptide-12 Acetate (Palmitoyl Hexapeptide-12 Acetate (171263-26-6 Free base)) 可以促进胶原蛋白、弹性蛋白和透明质酸的增殖。可用于改善皮肤含水量,增加真皮层厚度,减少细纹。
TP2486 Myristoyl Hexapeptide-16 Acetate

Myristoyl Hexapeptide-16 Acetate(959610-54-9 Free base)

Others Others
Myristoyl Hexapeptide-16 Acetate 被归类为一种蛋白质刺激肽,这意味着它可以帮助皮肤表面看起来更好,并且更能抵抗水分流失。
TP2494 Acetyl Hexapeptide-49 Acetate

Acetyl Hexapeptide-49 Acetate(1459205-54-9 Free base)

Others Others
Acetyl Hexapeptide-49 Acetate 可改善敏感皮肤因 PAR-2 诱导的促炎介质释放而出现的持续性疼痛和瘙痒的不适,此外还能恢复受损的屏障完整性。
TP2316 Myristoyl Hexapeptide-23 Acetate

Others Others
Myristoyl Hexapeptide-23 Acetate 有抗粉刺作用。
T81565 Palmitoyl hexapeptide-14

Palmitoyl hexapeptide-6

Palmitoyl hexapeptide-14(亦称为Palmitoyl hexapeptide-6)是一种生物活性肽,因其抗皱功能而常作为化妆品成分。
TP2382 Gastrin hexapeptide

Tyr-gly-trp-met-asp-phe-NH2,Gastrin C-terminal hexapeptide

Gastrin hexapeptide is a hexapeptide from porcine antral mucosa.
TP1253 Argireline

六胜肽,Acetyl hexapeptide-3,阿基瑞林

Others Others
Argireline (Acetyl hexapeptide-3) 是可渗透皮肤的、无毒的抗皱肽。它对神经肌肉接头处依赖 Ca2+的神经递质释放具有显著的抑制作用。它具有抗皱和抗衰老的活性。
T8953 Acetyl hexapeptide 38

Others Others
Acetyl hexapeptide 38 是一种乙酰化六肽,能显着刺激脂肪合成部位的使用,增加胸部或脸颊的体积,塑造完美身材
TP2384 Hexapeptide-10

Serilesine

Hexapeptide-10 is a synthetic peptide. It increases the synthesis of laminin V and α6-integrin to promote cell binding, with extraordinary visible skin restructuring and firming abilities.
TP2393 Neurotensin-related hexapeptide

Lant-6

Neurotensin-related hexapeptide exists in retinal ganglion cells and in their central projections in pigeons and may be utilized as a neuroactive substance by the central terminals of numerous retinal ganglion cells in birds.
TP2341 Hexapeptide-11

Peptamide 6,Fvapfp,Phe-val-ala-pro-phe-pro

Hexapeptide-11 is a novel proteostasis network modulator in human diploid fibroblasts.
T82205 Hexapeptide-3

Hexapeptide-3为生物活性肽,功能包括修复皮肤,已报道应用于化妆品成分。
T82203 Hexapeptide-42

Hexapeptide-42,一种具备生物活性的肽,常作为化妆品成分应用。
T64558 Hexapeptide 9

Hexapeptide 9 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64558。
T82204 Hexapeptide-33

Hexapeptide-33为一生物活性肽,报道显示其作为化妆品成分之用。
T82206 Hexapeptide-12

Hexapeptide-12为一生物活性肽,具抗衰老功能,现报道应用于化妆品成分中。
T34600 Secretin (1-6)

Secretin,N-terminal hexapeptide

Secretin (1-6) is the N-terminal part of secretin. It can produce vitro glucose-dependent insulin release induced by secretin.
T80200 Acetyl hexapeptide-49

Acetyl hexapeptide-49为生物活性肽,具抗敏感性能,应用于化妆品成分。
T81730 Myristoyl hexapeptide-16

Myristoyl hexapeptide-16,一种生物活性肽,具刺激睫毛生长功能,已报导为化妆品成分使用。
T81566 Palmitoyl hexapeptide-12

Palmitoyl hexapeptide-12,一种生物活性肽,具抗衰老(anti-aging)功能,常作为化妆品原料。
T83200 Acetyl hexapeptide-1

Melitane

Acetyl hexapeptide-1(Melitane)为一生物活性肽,具抗皱(anti-wrinkle)功能,已应用于化妆品成分中。
T83199 Acetyl hexapeptide-37

Acetyl hexapeptide-37是一种生物活性肽,具抗衰老(anti-aging)功能,常作为化妆品成分使用。
T64676 Melitane (Acetyl Hexapeptide-1) acetate

Melitane (Acetyl Hexapeptide-1) acetate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64676。
T22118 NQTrp

Microtubule Associated Cytoskeletal Signaling
NQTrp 是芳香萘醌-色氨酸杂交分子,可以抑制 tau 蛋白的聚集,具有抗淀粉样蛋白活性。NQTrp 对六肽 (41GCWMLY46,γD-crystallin 的 N 端)和全长 γD-crystallin 的体外聚集有抑制作用。
TP1250L Acetyl-PHF6 amide acetate(878663-43-5 freebase)

AcPHF6 acetate,Ac-VQIVYK-NH2 acetate

Others Others
Acetyl-PHF6 amide acetate(878663-43-5 freebase) (AcPHF6 acetate) 是一种 tau 衍生的六肽。
T31635 Enkephalin-met, lys(6)-

Met-enk-L,6-Lys-met-enkephalin

Enkephalin-met, lys(6)- is an opioid hexapeptide found in adrenal medulla.
T31568 DP 432

DP432,beta-Alanyl-Arg-Gly-Phe-Phe-Tyr-NH2,DP-432

DP 432 is an insulin hexapeptide fragment.
T25553 Jmv 332

Jmv-332,Jmv332

Jmv 332 is a cyclic analog of the C-terminal hexapeptide of CCK. It is a CCK/gastrin receptor agonist.
TP2350 RA X Peptide

RAX,RA-X,RA X

RA X Peptide is used as an antitumor cyclic hexapeptide.
T26028 RA VII

Methylether of TPC-A,RAVII,RA-VII

RA VII is used as an antitumor bicyclic hexapeptide of plant origin.
T24313 L 659874

L659874,L-659874

L 659874 is a cyclic hexapeptide. It is also a tachykinin antagonist.
T34654 Skf 107457

Skf107457,Skf-107457

Skf 107457 is a hexapeptide substrate analog with the scissile bond being replaced by a hydroxyethylene isostere.
T34507 San 201-456

Sandoz-201-456

San 201-456 is a cyclic hexapeptide somatostatin analog.
T24866 Tetrahydroechinocandin B

L 687,901,L-687901,L-687,901,L687,901,L 687901

Tetrahydroechinocandin B is a cyclic hexapeptide containing a fatty acyl side chain. It also inhibits 1,3-beta-D-glucan synthesis.
TP1250 Acetyl-PHF6 amide(TFA) (878663-43-5 free base)

Acetyl-PHF6 amide(TFA),AcPHF6 TFA,Ac-VQIVYK-NH2 TFA

Acetyl-PHF6 amide TFA is a tau derived hexapeptide.
T32440 L 363572

L363-572,L-363572,L-363-572,L363572,L 363-572

L 363572, a hexapeptide analog of MK 678, does not effect locomotor acitivity in rats.
T34174 Pseudobactin

Ferric pseudobactin

Pseudobactin is a linear hexapeptide fluorescent iron transport agent (siderophore) from plant growth promoter Pseudomonas B10.
T26192 SKF-107457

SKF 107457,Ala-Ala-Phepsi(CH(OH)CH2)Gly-Val-Val-OCH3

SKF-107457 is an HIV protease type 1 inhibitor. It is a hexapeptide substrate analog with the scissile bond being replaced by a hydroxy ethylene isostere.
T36032 Desotamide

Desotamide is a cyclic hexapeptide antibiotic originally isolated from Streptomyces. It is active against S. aureus, S. pneumoniae, and methicillin-resistant S. epidermidis (MRSE; MICs = 16, 12.5, and 32 μg/ml, respectively).
T75997 Acetyl-PHF6 amide TFA

Acetyl-PHF6 amide TFA (AcPHF6 TFA) 是 tau 衍生的六肽。
T76647 Acetyl-Amyloid β-Protein (1-6) amide

Acetyl-Amyloid β-Protein (1-6) amide 是一种具有潜在铜(II)结合位点的六肽,主要用于阿尔茨海默病及相关疾病的研究。
T40614 LCKLSL

LCKLSL, an N-terminal hexapeptide, acts as a competitive inhibitor of annexin A2 (AnxA2), effectively preventing the binding of tissue plasminogen activator (tPA) to AnxA2 while also inhibiting the generation of plasmin. In addition, LCKLSL exhibits anti-angiogenic properties.
T83102 Antiarrhythmic peptide (cattle atrium)

Antiarrhythmic peptide (cattle atrium)是一种具有保护作用的六肽,能对抗活性分子诱导的心律不齐。
T32372 Keenamide A

Keenamide A, a cytotoxic cyclic hexapeptide, exhibits significant activity towards the P-388, A-549, MEL-20, and HT-29 tumor cell lines, but was inactive against the D6 and W2 Plasmodium falciparum malarial clones.
T76092 Lys-Arg-Thr-Leu-Arg-Arg

Lys-Arg-Thr-Leu-Arg-Arg (KRTLRR) 是一种六肽。Lys-Arg-Thr-Leu-Arg-Arg 是EGF 受体蛋白激酶 C 的底物。Lys-Arg-Thr-Leu-Arg-Arg 可以用来测定蛋白激酶 C 的活性。
T24697 R 396

Acleu-asp-gln-trp-phe-glynh2,速激肽拮抗剂多肽

Neurokinin receptor GPCR/G Protein; Neuroscience
R 396 (Acleu-asp-gln-trp-phe-glynh2) 是一种线性六肽,也是一种 NK-2 速激肽受体拮抗剂。
T75904 PAR 4 (1-6) (TFA)

GYPGQV TFA (PAR 4 (1-6) TFA) 是一种六肽,作为蛋白酶激活受体 4 (PAR4) 片段,能特异性抑制PAR4。

化合物

Hexapeptide-10 Acetate
Cat.No: TP2384L
Synonym: Hexapeptide-10 Acetate(146439-94-3 Free base)
Target: Integrin
Hexapeptide-9 Acetate
Cat.No: TP2492
Synonym: Hexapeptide-9 Acetate(1228371-11-6 Free base)
Target: Others
Acetyl hexapeptide 38 Acetate
Cat.No: T8953L
Synonym: Acetyl hexapeptide 38 Acetate(1400634-44-7 free base)
Target: Others
Palmitoyl Hexapeptide-12 Acetate
Cat.No: TP2490
Synonym: Palmitoyl Hexapeptide-12 Acetate(171263-26-6 Free base)
Target: Others
Myristoyl Hexapeptide-16 Acetate
Cat.No: TP2486
Synonym: Myristoyl Hexapeptide-16 Acetate(959610-54-9 Free base)
Target: Others
Acetyl Hexapeptide-49 Acetate
Cat.No: TP2494
Synonym: Acetyl Hexapeptide-49 Acetate(1459205-54-9 Free base)
Target: Others
Myristoyl Hexapeptide-23 Acetate
Cat.No: TP2316
Synonym:
Target: Others
Palmitoyl hexapeptide-14
Cat.No: T81565
Synonym: Palmitoyl hexapeptide-6
Target:
Gastrin hexapeptide
Cat.No: TP2382
Synonym: Tyr-gly-trp-met-asp-phe-NH2,Gastrin C-terminal hexapeptide
Target:
Argireline
Cat.No: TP1253
Synonym: 六胜肽,Acetyl hexapeptide-3,阿基瑞林
Target: Others
Acetyl hexapeptide 38
Cat.No: T8953
Synonym:
Target: Others
Hexapeptide-10
Cat.No: TP2384
Synonym: Serilesine
Target:
Neurotensin-related hexapeptide
Cat.No: TP2393
Synonym: Lant-6
Target:
Hexapeptide-11
Cat.No: TP2341
Synonym: Peptamide 6,Fvapfp,Phe-val-ala-pro-phe-pro
Target:
Hexapeptide-3
Cat.No: T82205
Synonym:
Target:
Hexapeptide-42
Cat.No: T82203
Synonym:
Target:
Hexapeptide 9
Cat.No: T64558
Synonym:
Target:
Hexapeptide-33
Cat.No: T82204
Synonym:
Target:
Hexapeptide-12
Cat.No: T82206
Synonym:
Target:
Secretin (1-6)
Cat.No: T34600
Synonym: Secretin,N-terminal hexapeptide
Target:
Acetyl hexapeptide-49
Cat.No: T80200
Synonym:
Target:
Myristoyl hexapeptide-16
Cat.No: T81730
Synonym:
Target:
Palmitoyl hexapeptide-12
Cat.No: T81566
Synonym:
Target:
Acetyl hexapeptide-1
Cat.No: T83200
Synonym: Melitane
Target:
Acetyl hexapeptide-37
Cat.No: T83199
Synonym:
Target:
Melitane (Acetyl Hexapeptide-1) acetate
Cat.No: T64676
Synonym:
Target:
NQTrp
Cat.No: T22118
Synonym:
Target: Microtubule Associated
Acetyl-PHF6 amide acetate(878663-43-5 freebase)
Cat.No: TP1250L
Synonym: AcPHF6 acetate,Ac-VQIVYK-NH2 acetate
Target: Others
Enkephalin-met, lys(6)-
Cat.No: T31635
Synonym: Met-enk-L,6-Lys-met-enkephalin
Target:
DP 432
Cat.No: T31568
Synonym: DP432,beta-Alanyl-Arg-Gly-Phe-Phe-Tyr-NH2,DP-432
Target:
Jmv 332
Cat.No: T25553
Synonym: Jmv-332,Jmv332
Target:
RA X Peptide
Cat.No: TP2350
Synonym: RAX,RA-X,RA X
Target:
RA VII
Cat.No: T26028
Synonym: Methylether of TPC-A,RAVII,RA-VII
Target:
L 659874
Cat.No: T24313
Synonym: L659874,L-659874
Target:
Skf 107457
Cat.No: T34654
Synonym: Skf107457,Skf-107457
Target:
San 201-456
Cat.No: T34507
Synonym: Sandoz-201-456
Target:
Tetrahydroechinocandin B
Cat.No: T24866
Synonym: L 687,901,L-687901,L-687,901,L687,901,L 687901
Target:
Acetyl-PHF6 amide(TFA) (878663-43-5 free base)
Cat.No: TP1250
Synonym: Acetyl-PHF6 amide(TFA),AcPHF6 TFA,Ac-VQIVYK-NH2 TFA
Target:
L 363572
Cat.No: T32440
Synonym: L363-572,L-363572,L-363-572,L363572,L 363-572
Target:
Pseudobactin
Cat.No: T34174
Synonym: Ferric pseudobactin
Target:
SKF-107457
Cat.No: T26192
Synonym: SKF 107457,Ala-Ala-Phepsi(CH(OH)CH2)Gly-Val-Val-OCH3
Target:
Desotamide
Cat.No: T36032
Synonym:
Target:
Acetyl-PHF6 amide TFA
Cat.No: T75997
Synonym:
Target:
Acetyl-Amyloid β-Protein (1-6) amide
Cat.No: T76647
Synonym:
Target:
LCKLSL
Cat.No: T40614
Synonym:
Target:
Antiarrhythmic peptide (cattle atrium)
Cat.No: T83102
Synonym:
Target:
Keenamide A
Cat.No: T32372
Synonym:
Target:
Lys-Arg-Thr-Leu-Arg-Arg
Cat.No: T76092
Synonym:
Target:
R 396
Cat.No: T24697
Synonym: Acleu-asp-gln-trp-phe-glynh2,速激肽拮抗剂多肽
Target: Neurokinin receptor
PAR 4 (1-6) (TFA)
Cat.No: T75904
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T12448 Phomopsin A

Others Others
Phomopsin A is a cyclic hexapeptide mycotoxin isolated from the fungus Phomopsis leptostomiformis.
T27237 Echinocandin B

A-30912A,NSC 287461,A 30912A,A30912A,A22082

Echinocandin B is a cyclic hexapeptide echinocandin antibiotic from Aspergillus nidulans var. echinulatus . It attacks the cell wall of fungi by inhibiting beta-1,3-glucan synthesis.

天然产物

Phomopsin A
Cat.No: T12448
Synonym:
Target: Others
Echinocandin B
Cat.No: T27237
Synonym: A-30912A,NSC 287461,A 30912A,A30912A,A22082
Target:
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