Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11028 |
hDHODH-IN-4
DHODH-IN-5 |
Dehydrogenase | Metabolism |
hDHODH-IN-4 (DHODH-IN-5) 是一种有效的人二氢硼酸脱氢酶 (DHODH) 抑制剂,对人重组 DHODH 的 pIC50 为 7.8。hDHODH-IN-4 抑制麻疹病毒复制,pMIC50 为 8.8。 | |||
T11029 |
hDHODH-IN-5
DHODH-IN-7 |
Dehydrogenase | Metabolism |
hDHODH-IN-5 是人源二氢乳清酸脱氢酶的抑制剂 (hDHODH, IC50 = 0.91 μM)。 | |||
T11025 |
hDHODH-IN-3
DHODH-IN-2 |
Dehydrogenase | Metabolism |
hDHODH-IN-3 是人二氢乳清酸脱氢酶的抑制剂,pMIC50 值为 8.6。 hDHODH-IN-3 可以抑制麻疹病毒的复制。 | |||
T11546 |
hDHODH-IN-1
|
Dehydrogenase | Metabolism |
hDHODH-IN-1 是有效的人二氢乳清酸脱氢酶抑制剂, 显示出抗炎作用。 | |||
T11031 |
hDHODH-IN-7
DHODH-IN-9 |
Dehydrogenase | Metabolism |
hDHODH-IN-7 (DHODH-IN-9) 是一种含嗪的类似物,是一种人二氢乳清酸酯脱氢酶抑制剂。hDHODH-IN-7 具有抗病毒作用,pMIC50 为 7.4。 | |||
T64360 |
hDHODH-IN-8
|
Dehydrogenase | Metabolism |
hDHODH-IN-8 是人二氢乳清酸脱氢酶 (hDHODH) 的有效抑制剂,IC50 为 16 nM。 hDHODH-IN-8 具有强大的抗增殖活性和优异的水溶性。hDHODH-IN-8具有研究肿瘤疾病特别是淋巴瘤的潜力。 | |||
T11547 |
hDHODH-IN-2
|
Others | Others |
hDHODH-IN-2 is an analogue of the active metabolite of Leflunomide. hDHODH-IN-2 is a human dihydroorotate dehydrogenase (hDHODH) inhibitor with anti-inflammatory activity. | |||
T61226 |
hDHODH-IN-9
|
||
hDHODH-IN-9 (Compound 3k) is a highly potent inhibitor of hDHODH, exhibiting an IC50 of 0.34 μM. It displays significant cytotoxic activity against MCF-7 and A375 cells, while maintaining good selectivity. With its characteristics, hDHODH-IN-9 holds promise for cancer disease research [1]. | |||
T72948 |
hDHODH-IN-11
|
||
hDHODH-IN-11 是一种有效的人二氢旋转酸脱氢酶 (hDHODH) 抑制剂,其 IC50值为 7.2 nM。hDHODH-IN-11具有低细胞毒性。hDHODH-IN-11 可用于急性髓系白血病 (AML) 的研究。 | |||
T63037 | hDHODH-IN-10 | ||
hDHODH-IN-10 是一种选择性的、口服具有活力的、有效的 hDHODH 抑制剂 (IC50: 10.9 nM),能够与关键残基 Arg136 和 Gln47 形成氢键。hDHODH-IN-10 对癌细胞的增殖具有抑制作用,能够用于研究癌症(如 AML、结肠癌)。 | |||
T82223 | hDHODH-IN-13 | ||
hDHODH-IN-13是一种针对人二氢乳清酸脱氢酶(hDHODH)的抑制剂,具有IC50值为173.4 nM。该化合物可应用于炎症性肠病(IBD)的研究。 | |||
T78932 |
hDHODH-IN-12
|
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
hDHODH-IN-12是一种有效的DHODH抑制剂,IC50值为0.421 μM,DHODH作为嘧啶从头合成的限速酶,在(DNA/RNA Synthesis)DNA与RNA生成中扮演重要角色。hDHODH-IN-12位于人类线粒体内膜,展示了研究肺癌的潜力。 | |||
T40182 |
Ascochlorin A
Acremochlorin A |
||
Ascochlorin A is a novel and potent hDHODH inhibitor ( K D = 3.29 μM) for treatment of triple-negative breast cancer. |