Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15432 |
GSK256073
|
GPR; Others | Endocrinology/Hormones; GPCR/G Protein; Others |
GSK256073 是一种口服有活性的GPR109A 选择性激动剂,也是一种持久的人HCA2激动剂(pEC50:7.5) 。它能够减少脂降解,而显著改善葡萄糖稳态,对 2 型糖尿病和血脂异常具有潜在的研究价值。 | |||
T34573 |
SCH-900271
SCH 900271 |
AChR | Neuroscience |
SCH-900271是一种有效的尼古丁酸受体,用于治疗血脂异常,常用来研究混合性高脂血症和原发性高胆固醇血症。 | |||
T70849 | AZD-4121 | ||
AZD-4121 is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia. | |||
T70848 |
AZD-4121 tert-butylammonium
|
||
AZD-4121 tert-butylammonium is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia. |