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Cat. No. Product Name Target Signaling Pathways
T11120 Duocarmycin TM

DNA Alkylation; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Duocarmycin TM 是一种有抗肿瘤活性的抗生素,也是一种 DNA 烷化剂。
T23133 Pentamidine

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine 是抗微生物剂,会干扰 DNA 的生物合成。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它可用于冈比亚锥虫病,抗锑利什曼病和卡氏肺孢子虫肺炎的研究,有抗肿瘤活性,抗菌活性。
T11118 Duocarmycin SA

Others Others
Duocarmycin SA is an extremely potent cytotoxic agent and antitumor antibiotic that induces sequence-selective alkylation of duplex DNA, with an IC50 of 10 pM. It demonstrates synergistic cytotoxicity against glioblastoma multiforme (GBM) cells when combined with proton radiation in vitro.
T11338 Furamidine

DB75,NSC 305831

Others Others
Furamidine is also a selective and cell-permeable protein arginine methyltransferase 1 (PRMT1) inhibitor with an IC50 of 9.4 μM. Furamidine is selective for PRMT1 over PRMT5, PRMT6, and PRMT4 (CARM1) (IC50s of 166 μM, 283 μM, and >400 μM, respectively). Furamidine (DB75) is abisbenzamidine derivative and an antiparasite agent. Furamidine is a potent, reversible and competitive tyrosyl-DNA phosphodiesterase 1 (TDP-1) inhibitor. Inhibition of TDP-1 by Furamidine is effective both with single- and ...
T81640 NSC15520

NSC15520是一种小分子RPA抑制剂,特异性结合RPA的N端DNA结合域(DBD),阻断其与p53或RAD9的相互作用。它还能够抑制双链DNA(dsDNA)寡核苷酸的螺旋不稳定性,影响DNA复制、修复、重组及损伤反应信号。
T37218 N-methyl Mesoporphyrin IX

N-methyl Mesoporphyrin IX 是广泛使用的 G-quadruplex DNA 特异性荧光结合剂,能有效监测 Aβ 纤颤。N-methyl Mesoporphyrin IX 对 G-四链体 DNA 敏感,对双链体、三链体和单链形式的 DNA 没有反应。N-methyl Mesoporphyrin IX 需通过与 Aβ 组装体堆叠才能发出强荧光。同时 N-methyl Mesoporphyrin IX 是一种原位抑制剂,是体外和细胞内 Aβ 淀粉样蛋白生成的非原位监测器。

化合物

Duocarmycin TM
Cat.No: T11120
Synonym:
Target: DNA Alkylation, Antibiotic
Pentamidine
Cat.No: T23133
Synonym:
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Duocarmycin SA
Cat.No: T11118
Synonym:
Target: Others
Furamidine
Cat.No: T11338
Synonym: DB75,NSC 305831
Target: Others
NSC15520
Cat.No: T81640
Synonym:
Target:
N-methyl Mesoporphyrin IX
Cat.No: T37218
Synonym:
Target:
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